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GIPR [plasma membrane]
Stable Identifier
R-HSA-420132
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Gastric inhibitory polypeptide receptor, GIPR_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class B/2 (Secretin family receptors) (Homo sapiens)
Glucagon-type ligand receptors (Homo sapiens)
GIP receptor binds gastric inhibitory peptide (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
GIPR [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P48546 GIPR
Gene Names
GIPR
Chain
signal peptide:1-21, chain:22-466
Reference Genes
BioGPS Gene:2696 GIPR
COSMIC (genes):GIPR GIPR
CTD Gene:2696 GIPR
dbSNP Gene:2696 GIPR
ENSEMBL:ENSG00000010310 GIPR
ENSEMBL_homo_sapiens_GENE:ENSG00000010310.9 GIPR
HGNC:4271 GIPR
KEGG Gene (Homo sapiens):2696 GIPR
Monarch:2696 GIPR
NCBI Gene:2696 GIPR
OMIM:137241 GIPR
UCSC:P48546 GIPR
Reference Transcript
RefSeq:NM_001308418.1 GIPR
RefSeq:NM_000164.3 GIPR
Other Identifiers
11737205_a_at
16863326
208105_PM_at
208105_at
231291_PM_at
231291_at
2696
35589_at
35590_s_at
3836402
3836404
3836405
3836406
3836407
3836409
3836410
3836412
3836413
3836415
3836417
3836420
3836421
3836424
3836425
3836426
3836427
3836428
3836429
3836430
3836431
8029728
85939_at
A_23_P119395
GE484454
GO:0002029
GO:0004888
GO:0004930
GO:0005515
GO:0005886
GO:0006091
GO:0007165
GO:0007166
GO:0007186
GO:0007188
GO:0007189
GO:0007190
GO:0007204
GO:0007584
GO:0008528
GO:0009749
GO:0016020
GO:0016519
GO:0017046
GO:0023052
GO:0031018
GO:0032024
GO:0038192
GO:0043950
GO:0048678
GO:0048856
GO:0050796
GO:0051592
GO:0060089
GO:0070542
GO:0120022
Hs.192855.0.A1_3p_at
ILMN_2082005
PH_hs_0013304
TC19000651.hg
U39231_at
X81832_s_at
g4503998_3p_at
Participates
as an input of
GIP receptor binds gastric inhibitory peptide (Homo sapiens)
as a member of
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
as a component of
GIPR:GIP(52-93) [plasma membrane] (Homo sapiens)
Inferred To
GIPR [plasma membrane]
(Bos taurus)
GIPR [plasma membrane]
(Canis familiaris)
GIPR [plasma membrane]
(Gallus gallus)
GIPR [plasma membrane]
(Sus scrofa)
Gipr [plasma membrane]
(Mus musculus)
Gipr [plasma membrane]
(Rattus norvegicus)
gipr [plasma membrane]
(Xenopus tropicalis)
Cross References
RefSeq
NP_001295347.1
,
NP_000155.1
Guide to Pharmacology - Targets
248
OpenTargets
ENSG00000010310
ZINC - Substances
GIPR_HUMAN
ZINC target
P48546
PRO
P48546
PDB
7VAB
,
7FIN
,
4HJ0
,
6DKJ
,
2QKH
,
7RBT
,
7FIY
,
7DTY
,
7RA3
ZINC - Investigational
GIPR_HUMAN
GeneCards
P48546
HPA
ENSG00000010310-GIPR
Ensembl
ENSP00000305321
,
ENST00000304207
,
ENSP00000467494
,
ENSP00000263281
,
ENST00000590918
,
ENST00000263281
,
ENSG00000010310
Pharos - Targets
P48546
ZINC - Predictions - Purchasable
GIPR_HUMAN
Interactors (2)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P09681 GIP
6
GIP(22-153) [endoplasmic reticulum lumen]
(R-HSA-400512)
GIP(22-153) [secretory granule lumen]
(R-HSA-400526)
GIP(52-93) [secretory granule lumen]
(R-HSA-400483)
GIP(54-93) [extracellular region]
(R-HSA-400542)
GIP(1-153) [endoplasmic reticulum lumen]
(R-HSA-400470)
GIP(52-93) [extracellular region]
(R-HSA-400540)
0.618
3
UniProt:P01275 GCG
11
GCG(100-128) [extracellular region]
(R-HSA-400472)
ArgN-GCG(100-127) [extracellular region]
(R-HSA-400534)
GCG(1-180) [endoplasmic reticulum lumen]
(R-HSA-400456)
GCG(21-180) [endoplasmic reticulum lumen]
(R-HSA-381774)
GCG(21-180) [secretory granule lumen]
(R-HSA-421418)
ArgN-GCG(98-127) [secretory granule lumen]
(R-HSA-421419)
GLP-1 (7-37) [secretory granule lumen]
(R-HSA-421422)
GCG(146-178) [extracellular region]
(R-HSA-420211)
ArgN-GCG(98-127) [extracellular region]
(R-HSA-381699)
GLP-1 (7-37) [extracellular region]
(R-HSA-381636)
GCG(53-81) [extracellular region]
(R-HSA-163626)
0.558
2
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