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Opioid binds MOR
Stable Identifier
R-HSA-112042
Type
Reaction [binding]
Species
Homo sapiens
Compartment
extracellular region
,
plasma membrane
ReviewStatus
5/5
Locations in the PathwayBrowser
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Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (i) signalling events (Homo sapiens)
Opioid Signalling (Homo sapiens)
Opioid binds MOR (Homo sapiens)
General
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The layout of this reaction may differ from that in the pathway view due to the constraints in pathway layout
The binding of an opiate peptide to the mu opiate receptor stabilises the receptor conformation in a state of high affinity, both for the ligand itself, and for the G-protein.
Literature References
PubMed ID
Title
Journal
Year
7905839
Human mu opiate receptor. cDNA and genomic clones, pharmacologic characterization and chromosomal assignment
Wang, JB
,
Hawkins, AL
,
Persico, AM
,
Uhl, GR
,
Johnson, PS
,
Griffin, CA
FEBS Lett
1994
Participants
Input
Opioid peptide [extracellular region]
(Homo sapiens)
OPRM1 [plasma membrane]
(Homo sapiens)
Output
Opioid:MOR [plasma membrane]
(Homo sapiens)
Participates
as an event of
Opioid Signalling (Homo sapiens)
Orthologous Events
Opioid binds MOR (Bos taurus)
Opioid binds MOR (Canis familiaris)
Opioid binds MOR (Gallus gallus)
Opioid binds MOR (Mus musculus)
Opioid binds MOR (Rattus norvegicus)
Opioid binds MOR (Sus scrofa)
Opioid binds MOR (Xenopus tropicalis)
Authored
Jassal, B (2004-03-31)
Le Novere, N (2004-03-31)
Reviewed
Castagnoli, L (2008-11-06)
Created
Schmidt, EE (2004-04-06)
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