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WDR5 [nucleoplasm]
Stable Identifier
R-HSA-1629838
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
nucleoplasm
Synonyms
WD repeat-containing protein 5, BMP2-induced 3-kb gene protein, BIG3
Icon
Locations in the PathwayBrowser for interactor UniProt:Q14186
Expand all
Chromatin organization (Homo sapiens)
Chromatin modifying enzymes (Homo sapiens)
RMTs methylate histone arginines (Homo sapiens)
WDR5 binds Me2sR3-replicative histone H3 (Homo sapiens)
WDR5 [nucleoplasm] (Homo sapiens)
Developmental Biology (Homo sapiens)
Cardiogenesis (Homo sapiens)
EOMES, WDR5, KAT2A, and TBXT bind the MESP1 gene (Homo sapiens)
WDR5 [nucleoplasm] (Homo sapiens)
Gene expression (Transcription) (Homo sapiens)
Epigenetic regulation of gene expression (Homo sapiens)
Formation of WDR5-containing histone-modifying complexes (Homo sapiens)
Formation of the GCN5-ATAC complex (Homo sapiens)
WDR5 [nucleoplasm] (Homo sapiens)
Formation of the NSL complex (Homo sapiens)
WDR5 [nucleoplasm] (Homo sapiens)
Formation of the PCAF-ATAC complex (Homo sapiens)
WDR5 [nucleoplasm] (Homo sapiens)
Formation of the WRAD complex (Homo sapiens)
WDR5 [nucleoplasm] (Homo sapiens)
External Reference Information
External Reference
UniProt:P61964 WDR5
Gene Names
WDR5, BIG3
Chain
initiator methionine:, chain:2-334
Reference Genes
BioGPS Gene:11091 WDR5
COSMIC (genes):WDR5 WDR5
CTD Gene:11091 WDR5
dbSNP Gene:11091 WDR5
ENSEMBL:ENSG00000196363 WDR5
ENSEMBL_homo_sapiens_GENE:ENSG00000196363.10 WDR5
HGNC:12757 WDR5
KEGG Gene (Homo sapiens):11091 WDR5
Monarch:11091 WDR5
NCBI Gene:11091 WDR5
OMIM:609012 WDR5
UCSC:P61964 WDR5
Reference Transcript
RefSeq:NM_017588.2 WDR5
RefSeq:XM_005272163.1 WDR5
RefSeq:NM_052821.3 WDR5
Other Identifiers
11091
11718374_at
11718375_x_at
11718376_s_at
17090893
223308_PM_s_at
223308_s_at
225170_PM_at
225170_at
2724381
43017_at
43018_g_at
43410_at
43411_g_at
78481_at
8159111
89596_at
A_23_P32558
A_33_P3292417
GE55545
GO:0000122
GO:0000123
GO:0001501
GO:0003824
GO:0005515
GO:0005634
GO:0005654
GO:0005694
GO:0005856
GO:0005975
GO:0006094
GO:0006325
GO:0006351
GO:0006355
GO:0006357
GO:0016740
GO:0035064
GO:0035097
GO:0036211
GO:0042393
GO:0042800
GO:0043226
GO:0044545
GO:0044665
GO:0044666
GO:0045722
GO:0045815
GO:0045893
GO:0045995
GO:0048188
GO:0048856
GO:0051302
GO:0051571
GO:0051726
GO:0071339
GO:0072686
GO:0090043
GO:0140096
GO:0140672
HMNXSV003057386
Hs.13889.0.S1_3p_at
Hs.13889.0.S1_3p_x_at
Hs.323518.0.S1_3p_s_at
ILMN_1728626
ILMN_1737087
PH_hs_0028321
TC09000781.hg
Participates
as a member of
DCAF protein [nucleoplasm] (Homo sapiens)
as a component of
NSL (PHF20L1) [nucleoplasm] (Homo sapiens)
EOMES:WDR5:KAT2A:TBXT:MESP1 gene [nucleoplasm] (Homo sapiens)
NSL (PHF20) [nucleoplasm] (Homo sapiens)
GCN5-ATAC complex [nucleoplasm] (Homo sapiens)
PCAF-ATAC complex [nucleoplasm] (Homo sapiens)
ATAC complex [nucleoplasm] (Homo sapiens)
WDR5:Me2sR3-histone H3 [nucleoplasm] (Homo sapiens)
WRAD complex [nucleoplasm] (Homo sapiens)
as an input of
Formation of the NSL complex (Homo sapiens)
EOMES, WDR5, KAT2A, and TBXT bind the MESP1 gene (Homo sapiens)
Formation of the GCN5-ATAC complex (Homo sapiens)
Formation of the PCAF-ATAC complex (Homo sapiens)
WDR5 binds Me2sR3-replicative histone H3 (Homo sapiens)
Formation of the WRAD complex (Homo sapiens)
Inferred To
wu:fk47f04 [nucleoplasm]
(Danio rerio)
wdr5 [nucleoplasm]
(Dictyostelium discoideum)
wdr5 [nucleoplasm]
(Xenopus tropicalis)
swd3 [nucleoplasm]
(Schizosaccharomyces pombe)
Wdr5 [nucleoplasm]
(Mus musculus)
Wdr5 [nucleoplasm]
(Rattus norvegicus)
SWD3 [nucleoplasm]
(Saccharomyces cerevisiae)
WDR5 [nucleoplasm]
(Bos taurus)
WDR5 [nucleoplasm]
(Canis familiaris)
WDR5 [nucleoplasm]
(Gallus gallus)
WDR5 [nucleoplasm]
(Sus scrofa)
wds [nucleoplasm]
(Drosophila melanogaster)
wdr-5.1 [nucleoplasm]
(Caenorhabditis elegans)
Cross References
RefSeq
NP_438172.1
,
NP_060058.1
,
XP_005272220.1
Guide to Pharmacology - Targets
2831
OpenTargets
ENSG00000196363
ZINC - Substances
WDR5_HUMAN
ZINC target
P61964
PRO
P61964
PDB
6UCS
,
3N0D
,
6DAR
,
6OI1
,
8F1G
,
4O45
,
6U5Y
,
7AXS
,
6DAK
,
6E1Y
,
2H9M
,
7MBM
,
3UVL
,
6PGF
,
6UOZ
,
7AXQ
,
6U80
,
2H9L
,
6PG5
,
8Q1N
,
6PGD
,
8BB4
,
7CFQ
,
2O9K
,
6WJQ
,
6UFX
,
7CFP
,
2CO0
,
5EAP
,
6BYN
,
6PG3
,
6W5M
,
6PGA
,
3SMR
,
6PGC
,
8G3E
,
5SXM
,
4IA9
,
6DY7
,
6W5N
,
5EAL
,
7UD5
,
2G99
,
6OI2
,
8G3C
,
6DAS
,
4CY1
,
6W5I
,
7BCY
,
7MBN
,
2H9N
,
5EAR
,
6UHY
,
6E1Z
,
3P4F
,
6E22
,
6KIU
,
4EWR
,
6OI0
,
4QL1
,
3N0E
,
8E9F
,
8T5I
,
6U5M
,
3MXX
,
5EAM
,
5VFC
,
7JTP
,
6U8L
,
3UVM
,
7DNO
,
6DYA
,
6PGB
,
4ERY
,
6OI3
,
3UR4
,
2GNQ
,
6KIZ
,
4ERZ
,
7WVK
,
4Y7R
,
7AXX
,
4GM9
,
2H68
,
6KIV
,
6PWW
,
4CY2
,
7AXU
,
7UAS
,
4GM3
,
4ESG
,
2H13
,
2G9A
,
8DU4
,
6IAM
,
6PG8
,
7BED
,
6E23
,
3UVO
,
7JTO
,
2H9P
,
7AXP
,
3EG6
,
8F93
,
2H6K
,
3UVN
,
8BB3
,
3PSL
,
3EMH
,
7Q2J
,
4ES0
,
6UIK
,
5M23
,
6UJ4
,
4A7J
,
2H6Q
,
6U6W
,
6UIF
,
6UJJ
,
6KIW
,
6D9X
,
6PG9
,
7U9Y
,
4ERQ
,
6OFZ
,
6UJL
,
6KIX
,
4GMB
,
6DAI
,
6PG7
,
4GM8
,
6UJH
,
3UVK
,
6PWV
,
6UHZ
,
2CNX
,
6PG4
,
2H6N
,
8BB5
,
2H14
,
6PG6
,
6PGE
,
6U8O
,
8BB2
,
6U8B
,
5M25
GeneCards
P61964
HPA
ENSG00000196363-WDR5
Ensembl
ENSP00000351446
,
ENST00000358625
,
ENSG00000196363
Pharos - Targets
P61964
Orphanet
25037
ZINC - Predictions - Purchasable
WDR5_HUMAN
Interactors (87)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q03164 KMT2A
6
KMT2A [cytosol]
(R-HSA-9818584)
KMT2A(2719-3969) [cytosol]
(R-HSA-9818590)
KMT2A(1-2718) [cytosol]
(R-HSA-9818597)
KMT2A [nucleoplasm]
(R-HSA-1183223)
KMT2A(1-2718) [nucleoplasm]
(R-HSA-9818591)
KMT2A(2719-3969) [nucleoplasm]
(R-HSA-9818593)
0.953
13
UniProt:Q15291 RBBP5
1
RBBP5 [nucleoplasm]
(R-HSA-1629836)
0.948
15
UniProt:Q9UBL3 ASH2L
1
ASH2L [nucleoplasm]
(R-HSA-1629834)
0.942
15
UniProt:Q14686 NCOA6
1
NCOA6 [nucleoplasm]
(R-HSA-376414)
0.909
9
UniProt:Q9UMN6 KMT2B
5
KMT2B [cytosol]
(R-HSA-9818624)
KMT2B(2-2062) [cytosol]
(R-HSA-9818621)
KMT2B(2063-2715) [cytosol]
(R-HSA-9818626)
KMT2B(2063-2715) [nucleoplasm]
(R-HSA-9818623)
KMT2B(2-2062) [nucleoplasm]
(R-HSA-9818620)
0.896
8
UniProt:Q7Z3B3 KANSL1
1
KANSL1 [nucleoplasm]
(R-HSA-3321875)
0.885
12
UniProt:Q6ZW49 PAXIP1
1
PAXIP1 [nucleoplasm]
(R-HSA-5619395)
0.864
10
UniProt:O14686 KMT2D
1
KMT2D [nucleoplasm]
(R-HSA-1183219)
0.847
9
UniProt:Q9C005 DPY30
1
DPY30 [nucleoplasm]
(R-HSA-5669104)
0.812
8
UniProt:Q9NS73 MBIP
1
MBIP [nucleoplasm]
(R-HSA-3662291)
0.801
6
UniProt:O15047 SETD1A
1
SETD1A [nucleoplasm]
(R-HSA-3239027)
0.788
5
UniProt:Q03933 HSF2
0.781
7
UniProt:P51610 HCFC1
2
HCFC1 [nucleoplasm]
(R-HSA-1592209)
K48polyUb,K63polyUb-HCFC1 [nucleoplasm]
(R-HSA-5690821)
0.773
6
UniProt:Q9P0U4 CXXC1
1
CXXC1 [nucleoplasm]
(R-HSA-535610)
0.758
5
UniProt:Q2QGD7 ZXDC
0.743
5
UniProt:P68431 HIST1H3G
20
2xAcK-HIST1H3A [nucleoplasm]
(R-HSA-427507)
Ack-Me3K5-HIST1H3A [nucleoplasm]
(R-HSA-4551293)
AcK-Me3K10-HIST1H3A [nucleoplasm]
(R-HSA-4551291)
AcK-Me3K28-HIST1H3A [nucleoplasm]
(R-HSA-4551292)
Me2aR27-HIST1H3A [nucleoplasm]
(R-HSA-5229052)
Me2aR18-HIST1H3A [nucleoplasm]
(R-HSA-5229062)
Me2sR9-HIST1H3A [nucleoplasm]
(R-HSA-5211328)
Me2sR3-HIST1H3A [nucleoplasm]
(R-HSA-5218935)
AcK9,14-p-S10-HIST1H3A [nucleoplasm]
(R-HSA-8870893)
AcK14,18,79-p-S10-HIST1H3A [nucleoplasm]
(R-HSA-8871271)
AcK9,14,18-p-S10,T11-HIST1H3A [nucleoplasm]
(R-HSA-8871306)
AcK14,18-p-S10,T11-HIST1H3A [nucleoplasm]
(R-HSA-8871294)
AcK9,14,18,79-p-S10,T11-HIST1H3A [nucleoplasm]
(R-HSA-8865596)
AcK14,18-p-S10-HIST1H3A [nucleoplasm]
(R-HSA-8871295)
AcK14,18,79-p-T11-HIST1H3A [nucleoplasm]
(R-HSA-8871288)
AcK14,18-p-T11-HIST1H3A [nucleoplasm]
(R-HSA-8871299)
AcK14,18,79-p-S10,T11-HIST1H3A [nucleoplasm]
(R-HSA-8871286)
Me2K28-HIST1H3A [nucleoplasm]
(R-HSA-4754193)
MeK37-HIST1H3A [nucleoplasm]
(R-HSA-4722135)
MeK80-HIST1H3A [nucleoplasm]
(R-HSA-5649791)
0.74
11
UniProt:P54259 ATN1
1
ATN1 [nucleoplasm]
(R-HSA-6807083)
0.738
4
IntAct:EBI-15650351 H3TAIL
0.734
5
UniProt:Q9H9L4 KANSL2
1
KANSL2 [nucleoplasm]
(R-HSA-3321796)
0.734
4
UniProt:Q8IWI9 MGA
1
MGA [nucleoplasm]
(R-HSA-8953093)
0.725
4
UniProt:Q99496 RNF2
1
RNF2 [nucleoplasm]
(R-HSA-389119)
0.725
6
UniProt:Q9UPS6 SETD1B
1
SETD1B [nucleoplasm]
(R-HSA-5244714)
0.725
4
UniProt:Q9BTK6 PAGR1
1
PAGR1 [nucleoplasm]
(R-HSA-5619374)
0.725
5
UniProt:O15550 KDM6A
1
KDM6A [nucleoplasm]
(R-HSA-4754224)
0.708
6
UniProt:Q8NEZ4 KMT2C
1
KMT2C [nucleoplasm]
(R-HSA-1183224)
0.708
5
UniProt:O00255 MEN1
4
p-MEN1 [endoplasmic reticulum lumen]
(R-HSA-8956901)
MEN1 [endoplasmic reticulum lumen]
(R-HSA-8956785)
MEN1 [cytosol]
(R-HSA-5672315)
MEN1 [nucleoplasm]
(R-HSA-2186626)
0.708
4
UniProt:Q8NFC6 BOD1L1
1
BOD1L1 [nucleoplasm]
(R-HSA-8954547)
0.708
4
UniProt:Q9H7Z6 KAT8
1
KAT8 [nucleoplasm]
(R-HSA-3321802)
0.69
5
UniProt:P04637 TP53
20
Unfolded TP53 [cytosol]
(R-HSA-6813797)
TP53 [cytosol]
(R-HSA-8869337)
PolyUb-TP53 [nucleoplasm]
(R-HSA-6782509)
polySUMO2,3-K386-TP53 [nucleoplasm]
(R-HSA-2997661)
TP53 F341C [nucleoplasm]
(R-HSA-9726318)
TP53 G334V [nucleoplasm]
(R-HSA-9726126)
TP53 L330H [nucleoplasm]
(R-HSA-9726124)
TP53 A347T [nucleoplasm]
(R-HSA-9726339)
TP53 R337C [nucleoplasm]
(R-HSA-9726118)
TP53 L344P [nucleoplasm]
(R-HSA-9726075)
TP53 L344R [nucleoplasm]
(R-HSA-9726073)
TP53 R337H [nucleoplasm]
(R-HSA-9726169)
TP53 R337P [nucleoplasm]
(R-HSA-9726168)
TP53 L330P [nucleoplasm]
(R-HSA-9726136)
TP53 L348S [nucleoplasm]
(R-HSA-9726366)
TP53 R337L [nucleoplasm]
(R-HSA-9726163)
TP53 K351E [nucleoplasm]
(R-HSA-9726258)
TP53 F338I [nucleoplasm]
(R-HSA-9726358)
TP53 R342P [nucleoplasm]
(R-HSA-9726101)
TP53 L330R [nucleoplasm]
(R-HSA-9726133)
0.69
5
UniProt:Q9NS73-5 MBIP
0.666
4
UniProt:Q6PEV8 F199X
0.666
4
UniProt:Q9ULM3 YEATS2
1
YEATS2 [nucleoplasm]
(R-HSA-3321976)
0.643
3
UniProt:Q9P2R6 RERE
0.643
3
UniProt:Q9BYE7 PCGF6
1
PCGF6 [nucleoplasm]
(R-HSA-8953572)
0.643
4
UniProt:Q96EZ8 MCRS1
1
MCRS1 [nucleoplasm]
(R-HSA-3321849)
0.643
3
UniProt:O75528 TADA3
1
TADA3 [nucleoplasm]
(R-HSA-3322966)
0.643
3
UniProt:Q9Y5Z7 HCFC2
1
HCFC2 [nucleoplasm]
(R-HSA-9821232)
0.643
3
UniProt:Q8N488 RYBP
1
RYBP [nucleoplasm]
(R-HSA-8937975)
0.643
4
UniProt:Q96ES7 SGF29
1
SGF29 [nucleoplasm]
(R-HSA-3662279)
0.643
3
UniProt:Q13547 HDAC1
2
HDAC1 [nucleoplasm]
(R-HSA-205021)
monoSUMO1-K444,K476-HDAC1 [nucleoplasm]
(R-HSA-4616030)
0.643
3
UniProt:Q9BVI0 PHF20
2
p-S291-PHF20 [nucleoplasm]
(R-HSA-6805776)
PHF20 [nucleoplasm]
(R-HSA-3222239)
0.643
3
UniProt:O75461 E2F6
2
E2F6 [nucleoplasm]
(R-HSA-8953089)
p-S12-E2F6 [nucleoplasm]
(R-HSA-9007536)
0.643
4
UniProt:Q9HCK8 CHD8
1
CHD8 [nucleoplasm]
(R-HSA-3221598)
0.623
3
UniProt:Q8IYH5 ZZZ3
1
ZZZ3 [nucleoplasm]
(R-HSA-3662283)
0.623
3
UniProt:Q7Z434-1 MAVS
0.591
3
UniProt:O43823 AKAP8
0.576
3
UniProt:Q9D1P2
1
KAT8 [nucleoplasm]
(R-MMU-3321802)
0.564
2
UniProt:O15151 MDM4
5
PolyUb-MDM4 [nucleoplasm]
(R-HSA-6782502)
PolyUb,p-S342,S367,S403-MDM4 [nucleoplasm]
(R-HSA-6804938)
p-S346,S367,S403-MDM4 [nucleoplasm]
(R-HSA-349441)
p-S403-MDM4 [nucleoplasm]
(R-HSA-349461)
MDM4 [nucleoplasm]
(R-HSA-349430)
0.556
3
UniProt:A7MD48 SRRM4
0.556
3
UniProt:O76083-2 PDE9A
0.556
3
UniProt:Q9Y4F3 MARF1
0.556
6
UniProt:A2RRG2 A2RRG2
0.556
3
UniProt:Q9Y5X4 NR2E3
0.556
5
UniProt:Q9H891 Q9H891
0.556
3
UniProt:Q14204 DYNC1H1
3
DYNC1H1 [cytosol]
(R-HSA-380285)
DYNC1H1 [azurophil granule lumen]
(R-HSA-6799155)
DYNC1H1 [extracellular region]
(R-HSA-6806223)
0.556
3
UniProt:Q92794 KAT6A
3
KAT6A (1-1118) [nucleoplasm]
(R-HSA-5603260)
p-T369-KAT6A [nucleoplasm]
(R-HSA-6805633)
KAT6A [nucleoplasm]
(R-HSA-480310)
0.556
4
UniProt:Q9Y2D8 ADIP
0.556
3
UniProt:P10074 TZAP
0.556
3
UniProt:Q9UJX6 ANAPC2
2
ANAPC2 [cytosol]
(R-HSA-174229)
ANAPC2 [nucleoplasm]
(R-HSA-174141)
0.556
3
UniProt:Q6FHY5 Q6FHY5
0.556
3
UniProt:O00308 WWP2
1
WWP2 [cytosol]
(R-HSA-6807279)
0.556
3
UniProt:Q86V38 Q86V38
0.556
3
UniProt:Q96PG8 BBC3B
0.556
3
UniProt:Q92876 KLK6
0.556
3
IntAct:EBI-15662162 H3-8
0.544
2
UniProt:P01106 MYC
2
PolyUb-MYC [nucleoplasm]
(R-HSA-6783169)
MYC [nucleoplasm]
(R-HSA-188379)
0.536
2
UniProt:P58004 SESN2
1
SESN2 [cytosol]
(R-HSA-5629143)
0.527
2
UniProt:Q92769 HDAC2
2
monoSUMO1-K462-HDAC2 [nucleoplasm]
(R-HSA-4615958)
HDAC2 [nucleoplasm]
(R-HSA-205135)
0.527
2
UniProt:Q6UXN9 WDR82
1
WDR82 [nucleoplasm]
(R-HSA-9821474)
0.527
2
UniProt:P61513 RPL37A
1
RPL37A [cytosol]
(R-HSA-72468)
0.527
2
UniProt:O15294 OGT
2
OGT [nucleoplasm]
(R-HSA-3321845)
OGT [cytosol]
(R-HSA-9687814)
0.527
3
UniProt:Q06587 RING1
1
RING1 [nucleoplasm]
(R-HSA-389113)
0.527
3
UniProt:Q6ZSY5 PPR3F
0.527
2
UniProt:P19784 CSNK2A2
2
CSNK2A2 [nucleoplasm]
(R-HSA-6805065)
CSNK2A2 [cytosol]
(R-HSA-201721)
0.527
2
UniProt:Q9H8E8 KAT14
1
KAT14 [nucleoplasm]
(R-HSA-3301917)
0.527
2
UniProt:P49674 CSNK1E
2
CSNK1E [nucleoplasm]
(R-HSA-421306)
CSNK1E [cytosol]
(R-HSA-205877)
0.527
2
UniProt:Q6NZQ4 Paxip1
2
Paxip1 [nucleoplasm]
(R-MMU-5619398)
Paxip1 [nucleoplasm]
(R-MMU-5619395)
0.527
3
UniProt:Q9P2N6 KANSL3
1
KANSL3 [nucleoplasm]
(R-HSA-3321882)
0.527
2
UniProt:P83916 CBX1
1
CBX1 [nucleoplasm]
(R-HSA-9653629)
0.527
2
UniProt:Q969R5 L3MBTL2
2
L3MBTL2 [nucleoplasm]
(R-HSA-6804477)
polySUMO2-K675,K700-L3MBTL2 [nucleoplasm]
(R-HSA-6804480)
0.527
3
UniProt:Q13185 CBX3
1
CBX3 [nucleoplasm]
(R-HSA-427386)
0.527
3
UniProt:Q14186 TFDP1
1
TFDP1 [nucleoplasm]
(R-HSA-68652)
0.527
3
UniProt:Q13114 TRAF3
4
TRAF3 R118W [cytosol]
(R-HSA-5602321)
K48polyUb-TRAF3 [cytosol]
(R-HSA-936556)
TRAF3 [cytosol]
(R-HSA-914241)
K63polyUb-TRAF3 [cytosol]
(R-HSA-936402)
0.524
2
UniProt:Q9Y4K3 TRAF6
8
K48polyUb-TRAF6 [cytosol]
(R-HSA-6783233)
PolyUb-TRAF6 [cytosol]
(R-HSA-6782845)
TRAF6 [endosome membrane]
(R-HSA-450272)
K63polyUb-TRAF6 [endosome membrane]
(R-HSA-450227)
TRAF6 [cytosol]
(R-HSA-166366)
K63polyUb-TRAF6 [cytosol]
(R-HSA-2685681)
K63polyUb-TRAF6 [plasma membrane]
(R-HSA-936980)
TRAF6 [plasma membrane]
(R-HSA-936955)
0.524
2
UniProt:Q9NYB0 TERF2IP
1
TERF2IP [nucleoplasm]
(R-HSA-174873)
0.508
2
UniProt:Q9WTL8 Arntl
4
p-S-Arntl [nucleoplasm]
(R-MMU-508690)
Arntl [cytosol]
(R-MMU-508660)
Bmal1 [nucleoplasm]
(R-MMU-9634872)
Arntl [nucleoplasm]
(R-MMU-9769624)
0.508
2
UniProt:Q9H4Z2 ZNF335
1
ZNF335 [nucleoplasm]
(R-HSA-6810129)
0.462
2
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