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ADORA2A [Golgi membrane]
Stable Identifier
R-HSA-187668
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
Golgi membrane
Synonyms
Adenosine A2a receptor, AA2A_HUMAN
Locations in the PathwayBrowser for interactor UniProt:O15354 GPR37
Expand all
Signal Transduction (Homo sapiens)
Signaling by Receptor Tyrosine Kinases (Homo sapiens)
Signaling by NTRKs (Homo sapiens)
Signaling by NTRK1 (TRKA) (Homo sapiens)
Activation of TRKA receptors (Homo sapiens)
NGF-independant TRKA activation (Homo sapiens)
Ade-Rib binds AODORA2A and NTRK1,2 (Homo sapiens)
ADORA2A [Golgi membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P29274 ADORA2A
Gene Names
ADORA2A, ADORA2
Chain
chain:1-412
Reference Genes
BioGPS Gene:135 ADORA2A
COSMIC (genes):ADORA2A ADORA2A
CTD Gene:135 ADORA2A
dbSNP Gene:135 ADORA2A
ENSEMBL:ENSG00000128271 ADORA2A
HGNC:263 ADORA2A
KEGG Gene (Homo sapiens):135 ADORA2A
Monarch:135 ADORA2A
NCBI Gene:135 ADORA2A
OMIM:102776 ADORA2A
Reference Transcript
RefSeq:NM_001278499.1 ADORA2A
RefSeq:NM_001278497.1 ADORA2A
RefSeq:NM_000675.5 ADORA2A
RefSeq:NM_001278498.1 ADORA2A
RefSeq:NM_001278500.1 ADORA2A
Other Identifiers
11721939_a_at
11749942_a_at
135
205013_PM_s_at
205013_s_at
32114_s_at
3940102
3940103
3940104
3940105
3940106
3940107
3940111
3940112
3940113
3940114
3940115
8071899
A_23_P109436
A_24_P237270
A_33_P3214035
GE59944
GO:0000902
GO:0001609
GO:0001963
GO:0001973
GO:0001975
GO:0002376
GO:0003013
GO:0003674
GO:0004930
GO:0005515
GO:0005575
GO:0005622
GO:0005856
GO:0005882
GO:0005886
GO:0005887
GO:0006355
GO:0006464
GO:0006469
GO:0006810
GO:0006909
GO:0006915
GO:0006950
GO:0006954
GO:0006968
GO:0007155
GO:0007165
GO:0007186
GO:0007188
GO:0007189
GO:0007205
GO:0007267
GO:0007271
GO:0007417
GO:0007596
GO:0007600
GO:0007626
GO:0008015
GO:0008092
GO:0008150
GO:0008219
GO:0008283
GO:0008285
GO:0009058
GO:0009410
GO:0010035
GO:0012505
GO:0014049
GO:0014057
GO:0014061
GO:0014069
GO:0014074
GO:0015031
GO:0016020
GO:0016021
GO:0016192
GO:0019899
GO:0030154
GO:0030424
GO:0030425
GO:0030673
GO:0031000
GO:0031802
GO:0032230
GO:0032279
GO:0034641
GO:0035249
GO:0035810
GO:0035815
GO:0040011
GO:0040013
GO:0042311
GO:0042592
GO:0042734
GO:0042755
GO:0042802
GO:0043025
GO:0043116
GO:0043154
GO:0043226
GO:0043279
GO:0043524
GO:0044877
GO:0045211
GO:0045938
GO:0046636
GO:0048143
GO:0048786
GO:0048812
GO:0048856
GO:0050714
GO:0050728
GO:0050877
GO:0050896
GO:0051393
GO:0051881
GO:0051899
GO:0051924
GO:0051968
GO:0060079
GO:0060080
GO:0060134
GO:0098978
GO:0099055
GO:0099056
GO:0110148
GO:0110165
GO:1900273
GO:2000300
GO:2001235
HMNXSV003051303
ILMN_1807372
PH_hs_0022955
TC22001457.hg
X68486_at
g5921991_3p_a_at
Participates
as an input of
Ade-Rib binds AODORA2A and NTRK1,2 (Homo sapiens)
as a component of
Ade-Rib:ADORA2A:p-5Y-NTRK1,p-5Y-NTRK2 [Golgi membrane] (Homo sapiens)
Ade-Rib:ADORA2A:NTRK1,2 [Golgi membrane] (Homo sapiens)
Other forms of this molecule
ADORA2A [plasma membrane]
Cross References
RefSeq
NP_000666.2
,
NP_001265429.1
,
NP_001265426.1
,
NP_001265428.1
,
NP_001265427.1
ZINC - World Drugs
AA2AR_HUMAN
Guide to Pharmacology - Targets
19
OpenTargets
ENSG00000128271
ZINC - FDA approved
AA2AR_HUMAN
ZINC - Substances
AA2AR_HUMAN
ZINC target
P29274
ZINC - Biogenic
AA2AR_HUMAN
PRO
P29274
PDB
5NM2
,
3VG9
,
6LPK
,
6S0Q
,
5IU7
,
5NM4
,
3PWH
,
6WQA
,
6GT3
,
5IU4
,
5UIG
,
4EIY
,
5N2R
,
5MZJ
,
6PS7
,
5IUB
,
5MZP
,
5K2A
,
6JZH
,
4UG2
,
3REY
,
3UZC
,
5K2B
,
5UVI
,
6GDG
,
5IUA
,
6AQF
,
3QAK
,
5K2C
,
2YDO
,
3VGA
,
5WF5
,
5G53
,
5JTB
,
5IU8
,
6LPL
,
5NLX
,
5OLH
,
3EML
,
7ARO
,
6ZDR
,
5OLO
,
3RFM
,
6ZDV
,
5OLV
,
2YDV
,
4UHR
,
5OM1
,
5OLZ
,
3UZA
,
5OM4
,
5VRA
,
5K2D
,
6LPJ
,
6MH8
,
6S0L
,
7RM5
,
5OLG
,
5WF6
ZINC - Investigational
AA2AR_HUMAN
ZINC - Metabolites
AA2AR_HUMAN
HPA
ENSG00000128271-ADORA2A
GeneCards
P29274
Ensembl
ENSP00000336630
,
ENSP00000480012
,
ENSP00000481552
,
ENSP00000483102
,
ENST00000610595
,
ENST00000618076
,
ENST00000337539
,
ENSG00000128271
,
ENST00000611543
Pharos - Targets
P29274
ZINC - Predictions - Purchasable
AA2AR_HUMAN
Orphanet
22401
HMDB Protein
HMDBP01652
Interactors (13)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P29274 ADORA2A
2
ADORA2A [Golgi membrane]
(R-HSA-187668)
ADORA2A [plasma membrane]
(R-HSA-418934)
0.748
8
UniProt:Q7Z6G3 NECA2
0.71
6
UniProt:P21554 CNR1
1
CNR1 [plasma membrane]
(R-HSA-419411)
0.683
8
UniProt:Q99418 CYTH2
2
CYTH2 [cytosol]
(R-HSA-8847831)
CYTH2 [Golgi membrane]
(R-HSA-8847829)
0.634
6
UniProt:Q13107 USP4
1
USP4 [cytosol]
(R-HSA-5212663)
0.593
4
UniProt:Q5T9L3-1 WLS
0.589
3
UniProt:O15354 GPR37
1
GPR37 [plasma membrane]
(R-HSA-5333623)
0.581
3
UniProt:O43759-2 SYNGR1
0.556
3
UniProt:O15155 BET1
3
BET1 [Golgi membrane]
(R-HSA-6807743)
BET1 [transport vesicle]
(R-HSA-6808719)
BET1 [endoplasmic reticulum-Golgi intermediate compartment membrane]
(R-HSA-5688142)
0.556
3
UniProt:P14416 DRD2
1
DRD2 [plasma membrane]
(R-HSA-390816)
0.546
4
UniProt:P29275 ADORA2B
1
ADORA2B [plasma membrane]
(R-HSA-418898)
0.535
5
UniProt:P30542 ADORA1
1
ADORA1 [plasma membrane]
(R-HSA-418941)
0.518
4
UniProt:P31424-1 GRM5
0.463
3
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