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CYP3A5 [endoplasmic reticulum membrane]
Stable Identifier
R-HSA-211020
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
endoplasmic reticulum membrane
Synonyms
Cytochrome P450 3A5, CP35_HUMAN
Locations in the PathwayBrowser
Expand all
Metabolism (Homo sapiens)
Biological oxidations (Homo sapiens)
Aflatoxin activation and detoxification (Homo sapiens)
CYP1A2,3A4,3A5,2A13 oxidise AFB1 to AFXBO (Homo sapiens)
CYP1A2,3A4,3A5,2A13 [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A5 [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A4,5 hydroxylates AFB1 to AFQ1 (Homo sapiens)
CYP3A4,5 [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A5 [endoplasmic reticulum membrane] (Homo sapiens)
Phase I - Functionalization of compounds (Homo sapiens)
Cytochrome P450 - arranged by substrate type (Homo sapiens)
Xenobiotics (Homo sapiens)
CYP3A4 can N-demethylate loperamide (Homo sapiens)
Cytochrome P450 (CYPIIIA4 based) [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A5 [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A4,5 oxidise AFB1 to AFXBO (Homo sapiens)
Cytochrome P450 (CYP3A5 based) [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A5 [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A7 can 6beta-hydroxylate testosterone (Homo sapiens)
Cytochrome P450 (CYP3A7 based) [endoplasmic reticulum membrane] (Homo sapiens)
CYP3A5 [endoplasmic reticulum membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P20815 CYP3A5
Gene Names
CYP3A5
Chain
chain:1-502
Reference Genes
BioGPS Gene:1577 CYP3A5
COSMIC (genes):CYP3A5 CYP3A5
CTD Gene:1577 CYP3A5
dbSNP Gene:1577 CYP3A5
ENSEMBL:ENSG00000106258 CYP3A5
ENSEMBL_homo_sapiens_GENE:ENSG00000106258.16 CYP3A5
HGNC:2638 CYP3A5
KEGG Gene (Homo sapiens):1577 CYP3A5
Monarch:1577 CYP3A5
NCBI Gene:1577 CYP3A5
OMIM:605325 CYP3A5
UCSC:P20815 CYP3A5
Reference Transcript
RefSeq:NM_001190484.2 CYP3A5
RefSeq:NM_000777.4 CYP3A5
Other Identifiers
11721940_a_at
11721941_x_at
11760915_a_at
1577
17060287
205765_PM_at
205765_at
214234_PM_s_at
214234_s_at
243015_PM_at
243015_at
3063407
3063408
3063409
3063412
3063419
3063422
3063426
3063427
3063428
3063429
3063430
3063431
3063432
3063433
3063434
3063435
3063436
3063437
3063438
3063439
3063440
3063441
3063443
3063448
3063452
3063455
3063456
3063492
3063504
3063513
3063518
3063525
37124_i_at
37125_f_at
62681_at
70836_i_at
70838_r_at
8141328
A_23_P8801
A_24_P915256
A_24_P916916
A_33_P3249746
D00408_s_at
GE57519
GO:0002933
GO:0003824
GO:0004497
GO:0005506
GO:0005515
GO:0005783
GO:0005789
GO:0006629
GO:0006805
GO:0008202
GO:0008210
GO:0008401
GO:0009822
GO:0016020
GO:0016491
GO:0016705
GO:0016712
GO:0019825
GO:0020037
GO:0042178
GO:0042572
GO:0042573
GO:0043226
GO:0043231
GO:0046222
GO:0046872
GO:0050649
GO:0070330
GO:0070989
GO:0101020
HMNXSV003004318
HMNXSV003035397
HMNXSV003044217
Hs.269340.0.S1_3p_at
ILMN_1810942
TC07003079.hg
g4503230_3p_at
Participates
as a member of
CYP3A4,5 [endoplasmic reticulum membrane] (Homo sapiens)
Cytochrome P450 (CYP3A5 based) [endoplasmic reticulum membrane] (Homo sapiens)
CYP1A2,3A4,3A5,2A13 [endoplasmic reticulum membrane] (Homo sapiens)
as a candidate of
Cytochrome P450 (CYPIIIA4 based) [endoplasmic reticulum membrane] (Homo sapiens)
Cytochrome P450 (CYP3A7 based) [endoplasmic reticulum membrane] (Homo sapiens)
Inferred To
CYP3A5 [endoplasmic reticulum membrane]
(Bos taurus)
CYP3A5 [endoplasmic reticulum membrane]
(Canis familiaris)
CYP3A5 [endoplasmic reticulum membrane]
(Gallus gallus)
CYP3A5 [endoplasmic reticulum membrane]
(Mus musculus)
CYP3A5 [endoplasmic reticulum membrane]
(Rattus norvegicus)
CYP3A5 [endoplasmic reticulum membrane]
(Sus scrofa)
CYP3A5 [endoplasmic reticulum membrane]
(Xenopus tropicalis)
zgc:153269 [endoplasmic reticulum membrane]
(Danio rerio)
CYP3A [endoplasmic reticulum membrane]
(Danio rerio)
cyp3a4.1 [endoplasmic reticulum membrane]
(Xenopus tropicalis)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Bos taurus)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Canis familiaris)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Danio rerio)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Mus musculus)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Rattus norvegicus)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Sus scrofa)
Homologues of CYP3A5 [endoplasmic reticulum membrane]
(Xenopus tropicalis)
zgc:123110 [endoplasmic reticulum membrane]
(Danio rerio)
Cross References
RefSeq
NP_001177413.1
,
NP_000768.1
ZINC - World Drugs
CP3A5_HUMAN
Guide to Pharmacology - Targets
1338
OpenTargets
ENSG00000106258
ZINC - FDA approved
CP3A5_HUMAN
ZINC - Substances
CP3A5_HUMAN
ZINC target
P20815
PRO
P20815
PDB
5VEU
GeneCards
P20815
HPA
ENSG00000106258-CYP3A5
Ensembl
ENSG00000106258
,
ENSP00000222982
,
ENST00000646887
,
ENST00000222982
,
ENSP00000496704
,
ENST00000439761
,
ENSP00000401269
Pharos - Targets
P20815
ZINC - Predictions - Purchasable
CP3A5_HUMAN
Orphanet
19457
HMDB Protein
HMDBP01554
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P42858 HTT
1
HTT [nucleoplasm]
(R-HSA-9023590)
0.556
3
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