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ADRA1B [plasma membrane]
Stable Identifier
R-HSA-390661
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Alpha-1B adrenoceptor, RecName: Full=Alpha-1B adrenergic receptor; AltName: Full=Alpha 1B-adrenoreceptor; AltName: Full=Alpha 1B-adrenoceptor;
GN Name=ADRA1B;
OS Homo sapiens, ADA1B_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (12/13) signalling events (Homo sapiens)
Liganded G12/13-activating GPCR acts as a GEF for G12/13 (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (active). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (inactive). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Liganded G12/13-activating GPCRs bind inactive heterotrimeric G-protein G12/13 (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (inactive). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
The Ligand:GPCR:G12/13 complex dissociates (Homo sapiens)
GPCRs that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13:Heterotrimeric G-protein G12/13 (active). [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate G12/13 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Amine ligand-binding receptors (Homo sapiens)
Adrenoceptors (Homo sapiens)
ADRA1A,B,D bind ADR,NAd (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
ADRA1A,B,D:ADR,NAd [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
α1-agonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
α1-antagonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
α1-agonists bind ADRA1A,B,D (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
α1-agonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
α1-antagonists bind ADRA1A,B,D (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
α1-antagonists:ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1A,B,D [plasma membrane] (Homo sapiens)
ADRA1B [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P35368 ADRA1B
Gene Names
ADRA1B
Chain
chain:1-520
Reference Genes
BioGPS Gene:147 ADRA1B
COSMIC (genes):ADRA1B ADRA1B
CTD Gene:147 ADRA1B
dbSNP Gene:147 ADRA1B
ENSEMBL:ENSG00000170214 ADRA1B
ENSEMBL_homo_sapiens_GENE:ENSG00000170214.5 ADRA1B
HGNC:278 ADRA1B
KEGG Gene (Homo sapiens):147 ADRA1B
Monarch:147 ADRA1B
NCBI Gene:147 ADRA1B
OMIM:104220 ADRA1B
UCSC:P35368 ADRA1B
Reference Transcript
RefSeq:NM_000679.3 ADRA1B
Other Identifiers
11737368_at
147
16991705
207589_PM_at
207589_at
2837999
2838000
2838001
2838002
2838003
2838004
2838005
2838006
2838033
2838034
2838035
2838036
32983_at
8109612
A_23_P21929
A_23_P33326
GE80936
GO:0001996
GO:0003012
GO:0003013
GO:0004930
GO:0004935
GO:0004937
GO:0005515
GO:0005634
GO:0005635
GO:0005737
GO:0005886
GO:0005901
GO:0006937
GO:0007165
GO:0007186
GO:0007188
GO:0007200
GO:0007204
GO:0007267
GO:0016020
GO:0019229
GO:0023052
GO:0031965
GO:0035556
GO:0043226
GO:0043410
GO:0046982
GO:0055117
GO:0060089
GO:0071880
GO:0150099
HMNXSV003021821
HMNXSV003033117
ILMN_1679754
PH_hs_0025061
TC05000889.hg
g4501958_3p_at
Participates
as a member of
ADRA1A,B,D [plasma membrane] (Homo sapiens)
Inferred To
ser-5 [plasma membrane]
(Caenorhabditis elegans)
adra1b [plasma membrane]
(Xenopus tropicalis)
Adra1b [plasma membrane]
(Mus musculus)
Adra1b [plasma membrane]
(Rattus norvegicus)
TyrRII [plasma membrane]
(Drosophila melanogaster)
DopEcR [plasma membrane]
(Drosophila melanogaster)
TyrR [plasma membrane]
(Drosophila melanogaster)
ADRA1B [plasma membrane]
(Bos taurus)
ADRA1B [plasma membrane]
(Canis familiaris)
ADRA1B [plasma membrane]
(Gallus gallus)
ADRA1B [plasma membrane]
(Sus scrofa)
Homologues of ADRA1B [plasma membrane]
(Drosophila melanogaster)
Dmel\CG12290 [plasma membrane]
(Drosophila melanogaster)
zgc:103685 [plasma membrane]
(Danio rerio)
Cross References
RefSeq
NP_000670.1
ZINC - World Drugs
ADA1B_HUMAN
Guide to Pharmacology - Targets
23
OpenTargets
ENSG00000170214
ZINC - FDA approved
ADA1B_HUMAN
ZINC - Substances
ADA1B_HUMAN
ZINC target
P35368
ZINC - Biogenic
ADA1B_HUMAN
PRO
P35368
ZINC - Investigational
ADA1B_HUMAN
ZINC - Metabolites
ADA1B_HUMAN
GeneCards
P35368
HPA
ENSG00000170214-ADRA1B
Ensembl
ENSP00000306662
,
ENSG00000170214
,
ENST00000306675
Pharos - Targets
P35368
ZINC - Predictions - Purchasable
ADA1B_HUMAN
HMDB Protein
HMDBP07434
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P61073 CXCR4
1
CXCR4 [plasma membrane]
(R-HSA-2980772)
0.606
9
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