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GPR39 [plasma membrane]
Stable Identifier
R-HSA-443953
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
G-protein coupled receptor 39, GPR39_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Zinc is an agonist of GPR39 (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
GPR39 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:O43194 GPR39
Gene Names
GPR39
Chain
chain:1-453
Reference Genes
BioGPS Gene:2863 GPR39
COSMIC (genes):GPR39 GPR39
CTD Gene:2863 GPR39
dbSNP Gene:2863 GPR39
ENSEMBL:ENSG00000183840 GPR39
ENSEMBL_homo_sapiens_GENE:ENSG00000183840.8 GPR39
HGNC:4496 GPR39
KEGG Gene (Homo sapiens):2863 GPR39
Monarch:2863 GPR39
NCBI Gene:2863 GPR39
OMIM:602886 GPR39
UCSC:O43194 GPR39
Reference Transcript
RefSeq:NM_001508.2 GPR39
Other Identifiers
11739965_a_at
11739966_at
11755562_a_at
16885842
208600_PM_s_at
208600_s_at
229104_PM_s_at
229104_s_at
229105_PM_at
229105_at
2506569
2506571
2506572
2506573
2506606
2506607
2506608
2506609
2506610
2506611
2506613
2506615
2863
33142_at
8045336
A_23_P425240
A_23_P79155
GE569061
GO:0004930
GO:0005515
GO:0005886
GO:0007165
GO:0007186
GO:0016020
GO:0023052
GO:0046872
GO:0060089
HMNXSV003002606
Hs.85339.0.S1_3p_at
ILMN_1688768
PH_hs_0035856
TC02000865.hg
g4504096_3p_at
Participates
as a member of
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
as an input of
Zinc is an agonist of GPR39 (Homo sapiens)
as a component of
GPR39:Zn2+ [plasma membrane] (Homo sapiens)
Inferred To
GPR39 [plasma membrane]
(Bos taurus)
GPR39 [plasma membrane]
(Canis familiaris)
GPR39 [plasma membrane]
(Gallus gallus)
GPR39 [plasma membrane]
(Mus musculus)
GPR39 [plasma membrane]
(Sus scrofa)
LOC101732366 [plasma membrane]
(Xenopus tropicalis)
zgc:64187 [plasma membrane]
(Danio rerio)
Gpr39 [plasma membrane]
(Rattus norvegicus)
Cross References
RefSeq
NP_001499.1
Guide to Pharmacology - Targets
105
OpenTargets
ENSG00000183840
ZINC - Substances
GPR39_HUMAN
HPA
ENSG00000183840-GPR39
GeneCards
O43194
ZINC target
O43194
Ensembl
ENSP00000327417
,
ENST00000329321
,
ENSG00000183840
PRO
O43194
Pharos - Targets
O43194
ZINC - Predictions - Purchasable
GPR39_HUMAN
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P08908 HTR1A
1
HTR1A [plasma membrane]
(R-HSA-390971)
0.571
4
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