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RXFP1 [plasma membrane]
Stable Identifier
R-HSA-444834
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Relaxin receptor 1, RXFP1_HUMAN, LGR7
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Peptide ligand-binding receptors (Homo sapiens)
Relaxin receptors (Homo sapiens)
Relaxin receptor 1 binds relaxin 2 and 3 (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
RXFP1 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q9HBX9 RXFP1
Gene Names
RXFP1, LGR7
Chain
chain:1-757
Reference Genes
BioGPS Gene:59350 RXFP1
COSMIC (genes):RXFP1 RXFP1
CTD Gene:59350 RXFP1
dbSNP Gene:59350 RXFP1
ENSEMBL:ENSG00000171509 RXFP1
ENSEMBL_homo_sapiens_GENE:ENSG00000171509.16 RXFP1
HGNC:19718 RXFP1
KEGG Gene (Homo sapiens):59350 RXFP1
Monarch:59350 RXFP1
NCBI Gene:59350 RXFP1
OMIM:606654 RXFP1
UCSC:Q9HBX9 RXFP1
Reference Transcript
RefSeq:NM_021634.3 RXFP1
RefSeq:NM_001253728.1 RXFP1
RefSeq:NM_001253729.1 RXFP1
Other Identifiers
11748207_a_at
11750399_a_at
11750990_a_at
11761923_a_at
1552715_PM_a_at
1552715_a_at
16971910
231804_PM_at
231804_at
238206_PM_at
238206_at
2749507
2749508
2749520
2749523
2749524
2749525
2749526
2749528
2749529
2749530
2749531
2749532
2749533
2749534
2749535
2749536
2749537
2749540
2749541
2749542
2749543
2749544
2749545
2749546
2749547
2749548
2749549
59350
59756_at
79637_at
8098060
89447_at
A_14_P122746
A_23_P124534
A_23_P433050
GE61468
GE717026
GE80549
GO:0004930
GO:0005515
GO:0005886
GO:0007165
GO:0007186
GO:0007188
GO:0007189
GO:0007567
GO:0008528
GO:0009755
GO:0016020
GO:0022414
GO:0023052
GO:0030154
GO:0030198
GO:0036446
GO:0042562
GO:0046872
GO:0048856
GO:0060089
GO:0060427
GO:0060658
HMNXSV003021334
Hs.179243.0.A1_3p_at
Hs.209446.0.S2_3p_at
Hs2.209446.1.S1_3p_s_at
ILMN_1749150
PH_hs_0022861
Participates
as an input of
Relaxin receptor 1 binds relaxin 2 and 3 (Homo sapiens)
as a member of
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
as a component of
RXFP1:Relaxin-2,Relaxin-3 [plasma membrane] (Homo sapiens)
Inferred To
RXFP1 [plasma membrane]
(Bos taurus)
RXFP1 [plasma membrane]
(Canis familiaris)
RXFP1 [plasma membrane]
(Gallus gallus)
RXFP1 [plasma membrane]
(Mus musculus)
RXFP1 [plasma membrane]
(Rattus norvegicus)
RXFP1 [plasma membrane]
(Sus scrofa)
Rxfp1 [plasma membrane]
(Danio rerio)
rxfp1 [plasma membrane]
(Xenopus tropicalis)
Lgr4 [plasma membrane]
(Drosophila melanogaster)
Cross References
RefSeq
NP_001240658.1
,
NP_067647.2
,
NP_001240657.1
Guide to Pharmacology - Targets
351
OpenTargets
ENSG00000171509
GeneCards
Q9HBX9
HPA
ENSG00000171509-RXFP1
ZINC target
Q9HBX9
Ensembl
ENST00000471616
,
ENST00000343542
,
ENSP00000345889
,
ENST00000307765
,
ENSP00000303248
,
ENST00000470033
,
ENSG00000171509
,
ENSP00000434475
,
ENSP00000420712
PRO
Q9HBX9
Pharos - Targets
Q9HBX9
HMDB Protein
HMDBP02401
PDB
7TMW
,
2M7P
,
2JM4
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q08499-2 PDE4D
0.462
3
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