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KRAS [plasma membrane]
Stable Identifier
R-HSA-62719
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
p21A (K-Ras 2A), Transforming protein p21A, K-Ras 2A, Ki-Ras, c-K-ras
Locations in the PathwayBrowser
Expand all
Disease (Homo sapiens)
Diseases of signal transduction by growth factor receptors and second messengers (Homo sapiens)
Oncogenic MAPK signaling (Homo sapiens)
Signaling by moderate kinase activity BRAF mutants (Homo sapiens)
Activated MAP2Ks phosphorylate MAPKs downstream of moderate kinase activity BRAF mutants (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF:p-2S MAP2Ks:MAPKs:scaffold proteins [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF:p-2S MAP2Ks:p-T,Y MAPKs:scaffold proteins [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
Dissociation of moderate activity BRAF complexes (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF:p-2S MAP2Ks:p-T,Y MAPKs:scaffold proteins [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
Moderate kinase activity BRAF mutants bind RAS:GTP (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
p21 RAS:GTP:moderate kinase activity BRAF mutants [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
Moderate kinase activity BRAF mutants:RAS:GTP homo/heterodimerize (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
p21 RAS:GTP:moderate kinase activity BRAF mutants [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAF is phosphorylated downstream of moderate kinase activity BRAF mutants (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF complexes bind MAP2Ks and MAPKs (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF:MAP2Ks:MAPKs:scaffold proteins [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF complexes phosphorylate MAP2Ks (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF:MAP2Ks:MAPKs:scaffold proteins [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity p-RAF:p-2S MAP2Ks:MAPKs:scaffold proteins [plasma membrane] (Homo sapiens)
RAS:GTP:moderate kinase activity BRAF mutants:p-RAF:YWHAB [plasma membrane] (Homo sapiens)
RAS:GTP [plasma membrane] (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
Gene expression (Transcription) (Homo sapiens)
RNA Polymerase II Transcription (Homo sapiens)
Generic Transcription Pathway (Homo sapiens)
Transcriptional regulation by RUNX3 (Homo sapiens)
RUNX3 regulates p14-ARF (Homo sapiens)
Acetylated RUNX3 binds to BRD2 (Homo sapiens)
KRAS:GTP [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
Signal Transduction (Homo sapiens)
MAPK family signaling cascades (Homo sapiens)
MAPK1/MAPK3 signaling (Homo sapiens)
RAF/MAP kinase cascade (Homo sapiens)
RAS intrinsic GTPase activity hydrolyzes GTP to GDP (Homo sapiens)
RAS [plasma membrane] (Homo sapiens)
KRAS [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P01116 KRAS
Gene Names
KRAS, KRAS2, RASK2
Chain
chain:1-186, initiator methionine:, chain:2-186, propeptide:187-189
Reference Genes
BioGPS Gene:3845 KRAS
COSMIC (genes):KRAS KRAS
CTD Gene:3845 KRAS
dbSNP Gene:3845 KRAS
ENSEMBL:ENSG00000133703 KRAS
ENSEMBL_homo_sapiens_GENE:ENSG00000133703.14 KRAS
HGNC:6407 KRAS
KEGG Gene (Homo sapiens):3845 KRAS
Monarch:3845 KRAS
NCBI Gene:3845 KRAS
OMIM:190070 KRAS
UCSC:P01116 KRAS
Reference Transcript
RefSeq:XM_011520653.2 KRAS
RefSeq:NM_004985.4 KRAS
RefSeq:NM_033360.3 KRAS
RefSeq:XM_006719069.3 KRAS
Other Identifiers
11717962_x_at
11717963_a_at
11717964_a_at
11717965_s_at
16762399
1940_at
204009_PM_s_at
204009_s_at
204010_PM_s_at
204010_s_at
214352_PM_s_at
214352_s_at
231640_PM_at
231640_at
32159_at
3447860
3447862
3447864
3447865
3447866
3447867
3447868
3447869
3447870
3447871
3447872
3447873
3447874
3447879
3447880
3447884
3447885
3447886
3845
3958621
7961865
A_23_P306500
A_23_P306507
A_23_P45140
A_33_P3317815
GE61031
GO:0000139
GO:0000165
GO:0000166
GO:0001934
GO:0003824
GO:0003924
GO:0003925
GO:0005515
GO:0005525
GO:0005737
GO:0005739
GO:0005741
GO:0005783
GO:0005789
GO:0005794
GO:0005829
GO:0005886
GO:0005925
GO:0007010
GO:0007165
GO:0007265
GO:0008283
GO:0008542
GO:0009898
GO:0010467
GO:0010628
GO:0012501
GO:0012505
GO:0014009
GO:0016020
GO:0016601
GO:0016787
GO:0019003
GO:0021897
GO:0023052
GO:0030036
GO:0030154
GO:0030857
GO:0032228
GO:0035022
GO:0035914
GO:0036211
GO:0042802
GO:0043226
GO:0043495
GO:0043524
GO:0044877
GO:0048169
GO:0048856
GO:0048873
GO:0050877
GO:0051146
GO:0051402
GO:0060090
GO:0060252
GO:0060441
GO:0060509
GO:0098772
HMNXSV003005517
HMNXSV003016084
Hs.184050.0.S1_3p_a_at
Hs.184050.1.A1_3p_a_at
Hs.184050.4.A1_3p_at
ILMN_1652104
ILMN_1728071
M54968_at
PH_hs_0028364
PH_hs_0030345
TC12001314.hg
g4826811_3p_a_at
Participates
as a component of
KRAS:GTP [plasma membrane] (Homo sapiens)
as a member of
RAS [plasma membrane] (Homo sapiens)
Other forms of this molecule
S-Farn-Me-PalmS KRAS [plasma membrane]
p-Y32-S-Farn-Me-PalmS KRAS [plasma membrane]
KRAS A146T [plasma membrane]
KRAS K147E [plasma membrane]
KRAS K147T [plasma membrane]
KRAS V14G [plasma membrane]
KRAS K147N [plasma membrane]
KRAS A146V [plasma membrane]
KRAS A146S [plasma membrane]
KRAS A146P [plasma membrane]
KRAS P34R [plasma membrane]
KRAS P34L [plasma membrane]
KRAS G12A [plasma membrane]
KRAS G12R [plasma membrane]
KRAS G13V [plasma membrane]
KRAS G13S [plasma membrane]
KRAS G13C [plasma membrane]
KRAS G13R [plasma membrane]
KRAS G13A [plasma membrane]
KRAS K5N [plasma membrane]
KRAS G12S [plasma membrane]
KRAS Q61L [plasma membrane]
KRAS Q61K [plasma membrane]
KRAS Q61R [plasma membrane]
KRAS F156L [plasma membrane]
KRAS G12C [plasma membrane]
KRAS L19F [plasma membrane]
KRAS G12D [plasma membrane]
KRAS Q22E [plasma membrane]
KRAS K117N [plasma membrane]
KRAS Q22R [plasma membrane]
KRAS Q61H [plasma membrane]
KRAS V14I [plasma membrane]
KRAS G12V [plasma membrane]
KRAS D153V [plasma membrane]
KRAS G13D [plasma membrane]
KRAS T58I [plasma membrane]
KRAS G60R [plasma membrane]
KRAS D33E [plasma membrane]
KRAS Q22K [plasma membrane]
KRAS G60V [plasma membrane]
KRAS G60D [plasma membrane]
KRAS E63K [plasma membrane]
KRAS A59T [plasma membrane]
S-Farn-Me KRAS [endoplasmic reticulum membrane]
S-Farn-KRAS [endoplasmic reticulum membrane]
S-Farn-proKRAS [endoplasmic reticulum membrane]
proKRAS [cytosol]
Inferred To
KRAS [plasma membrane]
(Bos taurus)
KRAS [plasma membrane]
(Canis familiaris)
KRAS [plasma membrane]
(Gallus gallus)
KRAS [plasma membrane]
(Rattus norvegicus)
KRAS [plasma membrane]
(Sus scrofa)
RAS85D [plasma membrane]
(Drosophila melanogaster)
Kras [plasma membrane]
(Mus musculus)
HRAS [plasma membrane]
(Caenorhabditis elegans)
Cross References
RefSeq
XP_006719132.1
,
XP_011518955.1
,
NP_203524.1
,
NP_004976.2
Guide to Pharmacology - Targets
2824
OpenTargets
ENSG00000133703
ZINC - Substances
RASK_HUMAN
ZINC target
P01116
PRO
P01116
PDB
4EPV
,
4EPX
,
6CU6
,
6WGN
,
8EZG
,
7RSE
,
7RT3
,
1N4Q
,
6PGP
,
5UFQ
,
7ACA
,
5VPY
,
4M22
,
5VBM
,
6GOD
,
4LV6
,
5TB5
,
6MQN
,
6JTN
,
4PZZ
,
4OBE
,
7ACF
,
6GOF
,
6EPO
,
6JTP
,
6MNX
,
6WS2
,
7RP4
,
6PTW
,
7LC1
,
7R0Q
,
6GJ7
,
6FA2
,
3GFT
,
1N4P
,
5WHA
,
6PGO
,
1KZP
,
5OCO
,
7RP3
,
5VP7
,
5WHE
,
7Q9U
,
6VC8
,
8EPW
,
7R0N
,
5VQ6
,
8AQ7
,
6E6G
,
4M1W
,
5WLB
,
6CC9
,
1KZO
,
6EPP
,
7OO7
,
1D8E
,
6P8W
,
6P0Z
,
6E6F
,
7RT2
,
6BOF
,
6MS9
,
7YUZ
,
4LPK
,
4LYF
,
8I5E
,
6ZLI
,
4DSN
,
5VPI
,
8AZR
,
4Q02
,
5USJ
,
6JTO
,
6MQG
,
6XGV
,
5V9U
,
6VJJ
,
4M1Y
,
6H46
,
8STN
,
7F0W
,
5TAR
,
5V6S
,
8AZV
,
6F76
,
6BP1
,
8B6I
,
4EPT
,
7A1W
,
8AFB
,
7C40
,
7LGI
,
7A1Y
,
5XCO
,
5OCG
,
6EPL
,
7YCE
,
6GQY
,
7NY8
,
8AFC
,
7ACQ
,
7MDP
,
5UFE
,
5V9L
,
8DNJ
,
4DSO
,
6YR8
,
8G4H
,
7W5R
,
6V65
,
4LDJ
,
6ZL5
,
6ARK
,
7KFZ
,
8DNK
,
8JJS
,
6N2K
,
7LZ5
,
4TQ9
,
5WHB
,
7RP2
,
6OB2
,
5VQ8
,
7LC2
,
8EDY
,
4M1O
,
7RSC
,
4PZY
,
7OK4
,
5V6V
,
6XHA
,
1N4R
,
4LRW
,
8G4F
,
6QUU
,
5UQW
,
7YV1
,
5UK9
,
7MQU
,
4Q03
,
4TQA
,
6ASE
,
6GJ8
,
5VPZ
,
4LYJ
,
5WPM
,
8B00
,
8DNI
,
6O46
,
4Q01
,
5V9O
,
7C41
,
6OIM
,
7T47
,
7EYX
,
5US4
,
6MBU
,
1N4S
,
6W4E
,
5VQ0
,
5V71
,
5OCT
,
8B78
,
7OK3
,
6GOG
,
6CCH
,
7O70
,
7EWB
,
6EPN
,
4LYH
,
8EIE
,
6USX
,
6QUX
,
7ROV
,
6MTA
,
6GJ5
,
6H47
,
5YXZ
,
4M21
,
6CCX
,
6V6F
,
4EPW
,
4L8G
,
8G42
,
6TAM
,
7RT1
,
6V5L
,
8G9P
,
5YY1
,
6TAN
,
7A47
,
8G47
,
6GOE
,
6O4Y
,
5KYK
,
6OB3
,
6QUW
,
8CX5
,
8G9Q
,
8ECR
,
4NMM
,
6PTS
,
7R0M
,
6GOM
,
7U8H
,
4EPY
,
6B0Y
,
8AZZ
,
7T1F
,
7KMR
,
4LUC
,
6MBQ
,
8STM
,
6N2J
,
7RPZ
,
6USZ
,
6GQT
,
5MLA
,
7VVB
,
5WHD
,
5O2S
,
6B0V
,
6EPM
,
6GQX
,
6W4F
,
7TLK
,
6ASA
,
6P8Y
,
7EW9
,
4QL3
,
8AFD
,
5MLB
,
7A1X
,
5O2T
,
6YXW
,
6P8Z
,
6FA3
,
6O4Z
,
7SCX
,
7RT5
,
6UT0
,
7TLE
,
5F2E
,
5W22
,
6T5V
,
8AZX
,
6P8X
,
4WA7
,
6QUV
,
6T5B
,
8ONV
,
8EER
,
6O53
,
8AZY
,
6MBT
,
7ACH
,
6WS4
,
4M1S
,
6XHB
,
4EPR
,
6GQW
,
6M9W
,
7YCC
,
6FA4
,
7TLG
,
6GJ6
,
6FA1
,
6O51
,
5VQ1
,
4M1T
,
6T5U
,
6XGU
,
7KYZ
,
5VQ2
,
6O36
,
1D8D
,
7RT4
,
7SCW
,
8AQ5
,
6PQ3
,
7EWA
HPA
ENSG00000133703-KRAS
GeneCards
P01116
Ensembl
ENST00000685328
,
ENSP00000508921
,
ENSP00000256078
,
ENSP00000509238
,
ENST00000256078
,
ENST00000688940
,
ENSP00000308495
,
ENST00000311936
,
ENSG00000133703
Pharos - Targets
P01116
Orphanet
16312
HMDB Protein
HMDBP08526
Interactors (10)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P04049 RAF1
20
p-S338,Y340,Y341-RAF1 [cytosol]
(R-HSA-5624465)
p-S338-RAF1 [cytosol]
(R-HSA-5624469)
p-S621-RAF1 S259F [cytosol]
(R-HSA-9656124)
p-S621-RAF1 S257L [cytosol]
(R-HSA-9656121)
p-S621-RAF1 P261L [cytosol]
(R-HSA-9656106)
p-S621-RAF1 N262K [cytosol]
(R-HSA-9656101)
p-S621-RAF1 P261A [cytosol]
(R-HSA-9656103)
p-S621-RAF1 P261S [cytosol]
(R-HSA-9656113)
p-S621-RAF1 S259T [cytosol]
(R-HSA-9656130)
p-S621-RAF1 P261T [cytosol]
(R-HSA-9656115)
p-S621-RAF1 P261R [cytosol]
(R-HSA-9656110)
p-S621-RAF1 S259P [cytosol]
(R-HSA-9656127)
p-S621-RAF1 T260I [cytosol]
(R-HSA-9656136)
p-S621-RAF1 T260R [cytosol]
(R-HSA-9656139)
p-S621-RAF1 V263A [cytosol]
(R-HSA-9656148)
p-S621-RAF1 R256S [cytosol]
(R-HSA-9656119)
p-S621-RAF1 T491I [cytosol]
(R-HSA-9656143)
p-S621-RAF1 D486N [cytosol]
(R-HSA-9656088)
p-S621-RAF1 S427G [cytosol]
(R-HSA-9656134)
p-S621-RAF1 L613V [cytosol]
(R-HSA-9656098)
0.695
6
UniProt:Q99755 PIP5K1A
1
PIP5K1A [cytosol]
(R-HSA-1806260)
0.661
9
UniProt:Q96II5 Q96II5
0.556
3
UniProt:P50749 RASF2
0.544
2
UniProt:P61586 RHOA
6
RHOA [ficolin-1-rich granule membrane]
(R-HSA-6804971)
RHOA [secretory granule membrane]
(R-HSA-6804980)
RHOA [endoplasmic reticulum membrane]
(R-HSA-5672082)
RHOA [cytosol]
(R-HSA-194866)
RHOA [cell junction]
(R-HSA-2134503)
RHOA [plasma membrane]
(R-HSA-194510)
0.519
2
UniProt:O75915 ARL6IP5
1
ARL6IP5 [cytosol]
(R-HSA-2980942)
0.519
2
UniProt:P10398 ARAF
4
p-S299,S302,T452,T455,S582 ARAF [cytosol]
(R-HSA-5672646)
p-S299,S302,T452,T455,S582 ARAF [plasma membrane]
(R-HSA-5672648)
p-S582 ARAF [cytosol]
(R-HSA-5672681)
p-S214,S582 ARAF [cytosol]
(R-HSA-5672639)
0.483
2
UniProt:P28288 ABCD3
2
ABCD3 [cytosol]
(R-HSA-1456459)
ABCD3 [peroxisomal membrane]
(R-HSA-1456468)
0.483
2
UniProt:P15056 BRAF
20
BRAF(1-380)-MACF1(600-7388)fusion [cytosol]
(R-HSA-6802402)
p-BRAF(1-380)-MACF1(600-7388) fusion [cytosol]
(R-HSA-6802536)
BRAF E501G [cytosol]
(R-HSA-9651132)
BRAF D594N [cytosol]
(R-HSA-6802299)
BRAF D638E [cytosol]
(R-HSA-9651125)
BRAF G596R [cytosol]
(R-HSA-6802385)
BRAF D594V [cytosol]
(R-HSA-6802305)
BRAF G596V [cytosol]
(R-HSA-9651138)
BRAF G466E [cytosol]
(R-HSA-6802374)
BRAF D594G [cytosol]
(R-HSA-6802295)
BRAF L505H [cytosol]
(R-HSA-9648845)
BRAF F595L [cytosol]
(R-HSA-6802316)
BRAF L597V [cytosol]
(R-HSA-6802397)
BRAF G464E [cytosol]
(R-HSA-6802369)
BRAF N581D [cytosol]
(R-HSA-9651152)
BRAF E586K [cytosol]
(R-HSA-6802308)
BRAF V600K [cytosol]
(R-HSA-6802502)
BRAF A246P [cytosol]
(R-HSA-9651123)
BRAF G469V [cytosol]
(R-HSA-9648620)
BRAF T244P [cytosol]
(R-HSA-9651165)
0.483
3
ChEBI:16618 1-PHOSPHATIDYL-1D-MYO-INOSITOL 3,4,5-TRISPHOSPHATE
0.462
2
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