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CES1 [endoplasmic reticulum lumen]
Stable Identifier
R-HSA-2429659
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
endoplasmic reticulum lumen
Synonyms
Liver carboxylesterase 1 ecNumber3.1.1.1/ecNumber, EST1_HUMAN
Locations in the PathwayBrowser
Expand all
Drug ADME (Homo sapiens)
Aspirin ADME (Homo sapiens)
CES1,CES2 hydrolyze ASA- to ST (Homo sapiens)
CES1 trimer, CES2 [endoplasmic reticulum lumen] (Homo sapiens)
CES1 trimer [endoplasmic reticulum lumen] (Homo sapiens)
CES1 [endoplasmic reticulum lumen] (Homo sapiens)
Metabolism (Homo sapiens)
Biological oxidations (Homo sapiens)
Phase I - Functionalization of compounds (Homo sapiens)
CES1 trimer.CES2 hydrolyse COCN to BEG (Homo sapiens)
CES1 trimer, CES2 [endoplasmic reticulum lumen] (Homo sapiens)
CES1 trimer [endoplasmic reticulum lumen] (Homo sapiens)
CES1 [endoplasmic reticulum lumen] (Homo sapiens)
Metabolism of proteins (Homo sapiens)
Peptide hormone metabolism (Homo sapiens)
Metabolism of Angiotensinogen to Angiotensins (Homo sapiens)
CES1trimer hydrolyses ACEI pro-drugs to ACEIs (Homo sapiens)
CES1 trimer [endoplasmic reticulum lumen] (Homo sapiens)
CES1 [endoplasmic reticulum lumen] (Homo sapiens)
External Reference Information
External Reference
UniProt:P23141 CES1
Gene Names
CES1, CES2, SES1
Chain
signal peptide:1-17, chain:18-567
Reference Genes
BioGPS Gene:1066 CES1
COSMIC (genes):CES1 CES1
CTD Gene:1066 CES1
dbSNP Gene:1066 CES1
ENSEMBL:ENSG00000198848 CES1
ENSEMBL_homo_sapiens_GENE:ENSG00000198848.13 CES1
ENSEMBL_homo_sapiens_GENE:ENSG00000262243.5 CES1
HGNC:1863 CES1
KEGG Gene (Homo sapiens):1066 CES1
Monarch:1066 CES1
NCBI Gene:1066 CES1
OMIM:114835 CES1
UCSC:P23141 CES1
Reference Transcript
RefSeq:NM_001266.4 CES1
RefSeq:NM_001025194.1 CES1
RefSeq:NM_001025195.1 CES1
Other Identifiers
1066
11721638_s_at
16819152
16826639
17121404
209616_PM_s_at
209616_s_at
3661812
3661819
3661820
3661824
3661826
3661827
3661828
3661829
3661830
3661831
3661833
3661834
3661835
3661838
3661843
3661846
3661847
3661848
3661849
3661851
3661852
3661853
3661854
3661858
3692702
3692703
3692704
3692705
3692707
3692708
3692709
3692711
3692716
3692719
3692720
3692722
3692723
3692724
3692725
3692726
3692728
3692731
3692732
37203_at
8001457
8180234
ADDON000873.hg
A_23_P206733
A_33_P3241269
A_33_P3389704
GE57585
GE57586
GO:0003824
GO:0004771
GO:0005515
GO:0005737
GO:0005783
GO:0005788
GO:0005811
GO:0005829
GO:0006629
GO:0006695
GO:0008203
GO:0009636
GO:0010875
GO:0010887
GO:0016042
GO:0016192
GO:0016787
GO:0030154
GO:0030855
GO:0042632
GO:0043226
GO:0043691
GO:0047374
GO:0048856
GO:0051791
GO:0052689
GO:0070857
GO:0071397
GO:0071404
GO:0090122
GO:0090205
GO:0106435
GO:0120188
HMNXSV003037629
HMNXSV003043607
ILMN_1675386
ILMN_2359945
L07765_at
PH_hs_0027499
TC16001128.hg
TC16001572.hg
g688112_3p_at
Participates
as a component of
CES1 trimer [endoplasmic reticulum lumen] (Homo sapiens)
Other forms of this molecule
CES1 [lipid droplet]
Inferred To
Est-6 [endoplasmic reticulum lumen]
(Drosophila melanogaster)
cest-26 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
ges-1 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
cest-1.1 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
cryS [endoplasmic reticulum lumen]
(Dictyostelium discoideum)
Est-P [endoplasmic reticulum lumen]
(Drosophila melanogaster)
cest-2.2 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
GH05741 [endoplasmic reticulum lumen]
(Drosophila melanogaster)
zgc:153863 [endoplasmic reticulum lumen]
(Danio rerio)
CES5A [endoplasmic reticulum lumen]
(Canis familiaris)
cest-13 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
Jhe [endoplasmic reticulum lumen]
(Drosophila melanogaster)
Ghost homologue of CES1 [endoplasmic reticulum lumen]
(Xenopus tropicalis)
Dmel\CG12869 [endoplasmic reticulum lumen]
(Drosophila melanogaster)
Jhedup [endoplasmic reticulum lumen]
(Drosophila melanogaster)
Dmel\CG4382 [endoplasmic reticulum lumen]
(Drosophila melanogaster)
Ces1d [endoplasmic reticulum lumen]
(Mus musculus)
Ces1d [endoplasmic reticulum lumen]
(Rattus norvegicus)
cest-12 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
cest-2.1 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
D2 [endoplasmic reticulum lumen]
(Dictyostelium discoideum)
cest-2.3 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
cest-17 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
Homologues of CES1 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
Homologues of CES1 [endoplasmic reticulum lumen]
(Dictyostelium discoideum)
Homologues of CES1 [endoplasmic reticulum lumen]
(Drosophila melanogaster)
Homologues of CES1 [endoplasmic reticulum lumen]
(Gallus gallus)
Homologues of CES1 [endoplasmic reticulum lumen]
(Sus scrofa)
cest-1.2 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
CES1 [endoplasmic reticulum lumen]
(Bos taurus)
CES1 [endoplasmic reticulum lumen]
(Dictyostelium discoideum)
CES1 [endoplasmic reticulum lumen]
(Gallus gallus)
CES1 [endoplasmic reticulum lumen]
(Sus scrofa)
cest-16 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
cest-24 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
cest-19 [endoplasmic reticulum lumen]
(Caenorhabditis elegans)
Cross References
RefSeq
NP_001020365.1
,
NP_001257.4
,
NP_001020366.1
ZINC - World Drugs
EST1_HUMAN
Guide to Pharmacology - Targets
2592
OpenTargets
ENSG00000198848
ZINC - Substances
EST1_HUMAN
ZINC - Biogenic
EST1_HUMAN
ZINC target
P23141
PRO
P23141
PDB
8EOR
,
1MX1
,
1YAH
,
1YA4
,
4AB1
,
2HRQ
,
5A7G
,
3K9B
,
2HRR
,
2H7C
,
1YAJ
,
1YA8
,
5A7F
,
2DR0
,
1MX5
,
1MX9
,
2DQZ
,
5A7H
,
2DQY
ZINC - Investigational
EST1_HUMAN
ZINC - Metabolites
EST1_HUMAN
IntEnz
3.1.1.56
,
3.1.1.1
HPA
ENSG00000198848-CES1
GeneCards
P23141
Ensembl
ENSP00000353720
,
ENST00000422046
,
ENSP00000355193
,
ENST00000574513
,
ENST00000576783
,
ENSG00000262243
,
ENSG00000198848
,
ENSP00000460045
,
ENSP00000390492
,
ENSP00000461208
,
ENST00000571922
,
ENSP00000458586
,
ENST00000360526
,
ENST00000361503
Pharos - Targets
P23141
ZINC - Predictions - Purchasable
EST1_HUMAN
Orphanet
24405
HMDB Protein
HMDBP00497
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