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BRD1 [nucleoplasm]
Stable Identifier
R-HSA-3318450
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
nucleoplasm
Synonyms
Bromodomain-containing protein 1, BRD1_HUMAN, BRPF2
Locations in the PathwayBrowser
Expand all
Chromatin organization (Homo sapiens)
Chromatin modifying enzymes (Homo sapiens)
HATs acetylate histones (Homo sapiens)
KAT6A, KAT6B-containing ING5 complexes acetylate replicative histone H3 (Homo sapiens)
KAT6:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
Gene expression (Transcription) (Homo sapiens)
RNA Polymerase II Transcription (Homo sapiens)
Generic Transcription Pathway (Homo sapiens)
Transcriptional Regulation by TP53 (Homo sapiens)
Regulation of TP53 Activity (Homo sapiens)
Regulation of TP53 Activity through Acetylation (Homo sapiens)
AKT phosphorylates KAT6A (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
p-T369-KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
KAT6A acetylates TP53 (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:Ac-K120,K382,p-S15,S20-TP53 Tetramer [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:p-S15,S20-TP53 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
KAT6A and PML bind TP53 (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:p-S15,S20-TP53 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
MTA2-NuRD complex deacetylates TP53 (Homo sapiens)
BRD7:Ac-K382,p-S15,S20-TP53:EP300, KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:Ac-K120,K382,p-S15,S20-TP53 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:Ac-K120,K382,p-S15,S20-TP53 Tetramer [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:Ac-K120,p-S15,S20-TP53, BRD7:p-S15,S20-TP53:EP300 [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3):PML:Ac-K120,p-S15,S20-TP53 Tetramer [nucleoplasm] (Homo sapiens)
KAT6A:ING5:MEAF6:BRPF1,(2,3) [nucleoplasm] (Homo sapiens)
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
BRD1 [nucleoplasm] (Homo sapiens)
External Reference Information
External Reference
UniProt:O95696 BRD1
Gene Names
BRD1, BRL, BRPF2
Chain
chain:1-1058
Reference Genes
BioGPS Gene:23774 BRD1
COSMIC (genes):BRD1 BRD1
CTD Gene:23774 BRD1
dbSNP Gene:23774 BRD1
ENSEMBL:ENSG00000100425 BRD1
HGNC:1102 BRD1
KEGG:hsa:23774 BRD1
Monarch:23774 BRD1
NCBI Gene:23774 BRD1
OMIM:604589 BRD1
UCSC:O95696 BRD1
Reference Transcript
RefSeq:NM_001304809.1 BRD1
RefSeq:NM_001304808.1 BRD1
RefSeq:XM_017028716.1 BRD1
RefSeq:XM_017028717.1 BRD1
RefSeq:XM_017028715.1 BRD1
Other Identifiers
11731092_a_at
11731093_s_at
11748646_a_at
16936230
204520_PM_x_at
204520_x_at
215460_PM_x_at
215460_x_at
23774
3965315
3965316
3965317
3965318
3965319
3965320
3965321
3965322
3965326
3965327
3965328
3965332
3965338
3965339
3965340
3965342
3965347
3965354
3965355
3965356
3965357
39894_f_at
39895_r_at
41699_f_at
8076836
A_23_P166536
GE79901
GO:0000123
GO:0003824
GO:0005515
GO:0005634
GO:0005694
GO:0006325
GO:0006338
GO:0006355
GO:0006357
GO:0016607
GO:0016740
GO:0030425
GO:0035902
GO:0036408
GO:0036409
GO:0042393
GO:0043204
GO:0043226
GO:0043249
GO:0043995
GO:0043996
GO:0043997
GO:0045648
GO:0046872
GO:0050793
GO:0051602
GO:0060090
GO:0070776
GO:0140096
GO:0140566
GO:1903706
HMNXSV003022918
HMNXSV003028782
Hs.127950.1.A1_3p_a_at
ILMN_1730019
PH_hs_0024160
TC22000902.hg
g11321641_3p_x_at
Participates
as a candidate of
BRPF1, (BRPF2, 3) [nucleoplasm] (Homo sapiens)
Inferred To
Brd1 [nucleoplasm]
(Mus musculus)
Brd1 [nucleoplasm]
(Rattus norvegicus)
lin-49 [nucleoplasm]
(Caenorhabditis elegans)
nto1 [nucleoplasm]
(Schizosaccharomyces pombe)
brd1a [nucleoplasm]
(Danio rerio)
BRD1 [nucleoplasm]
(Bos taurus)
BRD1 [nucleoplasm]
(Canis familiaris)
BRD1 [nucleoplasm]
(Dictyostelium discoideum)
BRD1 [nucleoplasm]
(Drosophila melanogaster)
BRD1 [nucleoplasm]
(Gallus gallus)
BRD1 [nucleoplasm]
(Sus scrofa)
brd1 [nucleoplasm]
(Xenopus tropicalis)
Cross References
RefSeq
NP_001291737.1
,
XP_016884204.1
,
NP_001291738.1
,
XP_016884206.1
,
XP_016884205.1
Guide to Pharmacology - Targets
2724
OpenTargets
ENSG00000100425
ENSEMBL
ENSP00000216267
,
ENSP00000384076
,
ENST00000457780
,
ENST00000216267
,
ENSP00000410042
,
ENSP00000385858
,
ENST00000404760
,
ENST00000404034
HPA
ENSG00000100425-BRD1
ZINC - Substances
BRD1_HUMAN
ZINC target
O95696
PRO
O95696
Pharos - Targets
O95696
GlyGen
O95696
ZINC - Predictions - Purchasable
BRD1_HUMAN
PDB
5PSM
,
5PS6
,
5PTS
,
5PSB
,
5PTY
,
5PUB
,
5PVK
,
5PS8
,
5PW6
,
5PO3
,
5PV3
,
5PSW
,
5PVG
,
5PW3
,
5PTO
,
5PTW
,
5PV7
,
5PTG
,
5PUO
,
5PP2
,
5POV
,
5PPH
,
4Z02
,
5PO5
,
5POE
,
5PPN
,
5PQQ
,
5PPV
,
5POJ
,
5PPD
,
5PR6
,
5PPQ
,
5PRB
,
5PSS
,
5PQJ
,
5PNY
,
5PPZ
,
5PS2
,
5PR7
,
5PRU
,
5PRM
,
5PT5
,
5PU5
,
5PSC
,
5PSJ
,
5PTZ
,
5PUC
,
5PVL
,
5PUL
,
5PVU
,
5PRW
,
5PUV
,
5PUR
,
5PVH
,
5PVR
,
5PU1
,
5PU9
,
5PTH
,
5PPE
,
3RCW
,
5PP8
,
5PPA
,
7D0P
,
5PQN
,
5POQ
,
5PWB
,
5PO0
,
5POK
,
5PQU
,
2LQ6
,
5PQ3
,
5PQK
,
5PNZ
,
5PQD
,
5PRQ
,
5N49
,
5PT1
,
5PQV
,
5PQ8
,
5PW5
,
5PRY
,
5PTJ
,
5PV6
,
5PQL
,
5PRD
,
5PR5
,
5PS5
,
2L43
,
5PSX
,
5PTV
,
5PSV
,
5PTB
,
5PSD
,
5PW2
,
5PVI
,
5PUD
,
5PVM
,
5PUN
,
5PW9
,
5PUX
,
5PP1
,
5POG
,
7D0Q
,
5PO7
,
5PPP
,
5POU
,
6MAK
,
6IN2
,
5PS1
,
5PQP
,
5PPU
,
5PPJ
,
5POY
,
5PTR
,
5PSR
,
5PQX
,
5PRG
,
5PPT
,
5PUU
,
5PSL
,
5PU4
,
5PRZ
,
5PQM
,
5PO2
,
3LYI
,
5PSY
,
5PT8
,
5PVT
,
5PSE
,
5PVJ
,
5PVQ
,
5PU8
,
5PU0
,
5PUE
,
5PVN
,
5PV0
,
5PVX
,
5PUA
,
5PUY
,
5POA
,
5POP
,
5PPG
,
5PP7
,
5POD
,
5PO4
,
5PPM
,
5PR2
,
5PQ7
,
5PRP
,
5PPC
,
5PT4
,
5PQT
,
5PRT
,
5PQY
,
5PRA
,
5PQ2
,
5PPY
,
5PRH
,
5PW4
,
5PUK
,
5PSZ
,
5PTC
,
5PV5
,
5PSU
,
5PRE
,
5PQZ
,
5PS4
,
5PT0
,
5PSF
,
5PTU
,
5PTK
,
5POL
,
5PVC
,
5PUF
,
7LH9
,
5PW8
,
5PW1
,
5PV2
,
5PPO
,
5POF
,
5POT
,
5PNX
,
5POC
,
5PP4
,
5POO
,
5PSQ
,
5PPX
,
5PQF
,
5PS0
,
6MAJ
,
5PTQ
,
5PSI
,
2KU3
,
5PRI
,
5PPS
,
5PPL
,
5PP9
,
5PQS
,
5PQC
,
5PVS
,
5PUT
,
5PRF
,
5PRS
,
5PSO
,
5PSG
,
5PT7
,
5PU7
,
5PTA
,
5PTL
,
5PT9
,
5POM
,
5PVD
,
5PUZ
,
5PVW
,
5PUG
,
5PVP
,
5PV9
,
5PUQ
,
5PQ1
,
5PP6
,
5PO6
,
5POS
,
7D0R
,
7D0S
,
5PQA
,
5FG6
,
5PRO
,
5PQG
,
5PR1
,
5PQ6
,
5PU3
,
5PT3
,
5POX
,
5PPI
,
5PRJ
,
5PR9
,
5PQ5
,
5PS7
,
5PST
,
5PTT
,
5PSK
,
5PTE
,
5PUM
,
5PRK
,
5PW7
,
5PSA
,
5PS9
,
5PV8
,
5PTM
,
5AME
,
5PV4
,
5PVA
,
5PUH
,
5PV1
,
5PVY
,
5PTX
,
5PVE
,
5PW0
,
5PPF
,
5POH
,
5PPB
,
5PPR
,
5PP3
,
5POB
,
5POW
,
5PO8
,
5PR0
,
5PON
,
5PWA
,
5PO1
,
5GK9
,
5PQE
,
5PS3
,
5PQR
,
5PR8
,
5PQH
,
5PPW
,
5PSP
,
5PUJ
,
5PRV
,
5PT6
,
5PVV
,
5PTF
,
5PRL
,
5PUW
,
5PU2
,
5PRX
,
5PUS
,
5PSN
,
5PTN
,
5AMF
,
5PU6
,
5PVB
,
5PUI
,
5PVZ
,
5PVF
,
5PVO
,
5PUP
,
5PQ0
,
5PP5
,
5POI
,
7D0O
,
5POR
,
5PO9
,
5PQO
,
5PP0
,
5PQW
,
5PSH
,
5PR4
,
5POZ
,
5PQ4
,
5PPK
,
5PQI
,
5PQ9
,
5PRR
,
5PQB
,
5PT2
Interactors (4)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q9UBB9 TFIP11
1
TFIP11 [nucleoplasm]
(R-HSA-8869310)
0.556
3
UniProt:Q9NRD5 PICK1
2
PICK1 [plasma membrane]
(R-HSA-416989)
PICK1 [endocytic vesicle membrane]
(R-HSA-417017)
0.556
3
UniProt:Q9UGI0 ZRANB1
1
ZRANB1 [cytosol]
(R-HSA-6781939)
0.556
3
UniProt:P62258 YWHAE
1
YWHAE [cytosol]
(R-HSA-194368)
0.483
2
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