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KISS1R [plasma membrane]
Stable Identifier
R-HSA-388974
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
RecName: Full=KiSS-1 receptor; Short=KiSS-1R; AltName: Full=Kisspeptins receptor; AltName: Full=Metastin receptor; AltName: Full=G-protein coupled receptor 54; AltName: Full=Hypogonadotropin-1; Short=hOT7T175;
GN Name=KISS1R; Synonyms=AXOR12, GPR54, OT7T175;
OS Homo sapiens, KISSR_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (q) signalling events (Homo sapiens)
Liganded Gq-activating GPCRs bind inactive heterotrimeric Gq (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
Liganded Gq/11-activating GPCRs act as GEFs for Gq/11 (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gq complex dissociates (Homo sapiens)
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11:Heterotrimeric G-protein Gq (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gq/11 [plasma membrane] (Homo sapiens)
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Peptide ligand-binding receptors (Homo sapiens)
The Kiss receptor GPR54 binds kisspeptin (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
KISS1R [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q969F8 KISS1R
Gene Names
KISS1R, AXOR12, GPR54
Chain
chain:1-398
Reference Genes
BioGPS Gene:84634 KISS1R
COSMIC (genes):KISS1R KISS1R
CTD Gene:84634 KISS1R
dbSNP Gene:84634 KISS1R
ENSEMBL:ENSG00000116014 KISS1R
ENSEMBL_homo_sapiens_GENE:ENSG00000116014.10 KISS1R
HGNC:4510 KISS1R
KEGG Gene (Homo sapiens):84634 KISS1R
Monarch:84634 KISS1R
NCBI Gene:84634 KISS1R
OMIM:604161 KISS1R
UCSC:Q969F8 KISS1R
Reference Transcript
RefSeq:NM_032551.4 KISS1R
Other Identifiers
11740202_at
16856307
242517_PM_at
242517_at
3815269
3815270
3815271
3815272
3815274
3815275
3815276
3815277
70594_at
8024070
84634
A_14_P107164
A_23_P101761
A_33_P3231357
GE87794
GO:0004930
GO:0005515
GO:0005886
GO:0005929
GO:0007165
GO:0007186
GO:0007218
GO:0008188
GO:0008528
GO:0009986
GO:0016020
GO:0023052
GO:0043226
GO:0043231
GO:0060089
HMNXSV003029048
Hs.208229.0.A1_3p_at
ILMN_1673521
PH_hs_0029427
TC19000022.hg
Participates
as an input of
The Kiss receptor GPR54 binds kisspeptin (Homo sapiens)
as a member of
GPCRs that activate Gq/11 [plasma membrane] (Homo sapiens)
as a component of
KISS1R:KISS1(68-121) [plasma membrane] (Homo sapiens)
Inferred To
AstA-R2 [plasma membrane]
(Drosophila melanogaster)
npr-14 [plasma membrane]
(Caenorhabditis elegans)
Kiss1r [plasma membrane]
(Mus musculus)
Kiss1r [plasma membrane]
(Rattus norvegicus)
CG 13579 [plasma membrane]
(Drosophila melanogaster)
si:ch211-157p22.8 [plasma membrane]
(Danio rerio)
Homologues of KISS1R [plasma membrane]
(Drosophila melanogaster)
KISS1R [plasma membrane]
(Bos taurus)
KISS1R [plasma membrane]
(Canis familiaris)
KISS1R [plasma membrane]
(Sus scrofa)
Cross References
RefSeq
NP_115940.2
ZINC - World Drugs
KISSR_HUMAN
Guide to Pharmacology - Targets
266
OpenTargets
ENSG00000116014
ZINC - FDA approved
KISSR_HUMAN
ZINC - Substances
KISSR_HUMAN
ZINC target
Q969F8
PRO
Q969F8
PDB
7YQE
GeneCards
Q969F8
HPA
ENSG00000116014-KISS1R
Ensembl
ENSP00000234371
,
ENSG00000116014
,
ENST00000234371
Pharos - Targets
Q969F8
Orphanet
16307
ZINC - Predictions - Purchasable
KISSR_HUMAN
HMDB Protein
HMDBP07764
Interactors (1)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:P67775 PPP2CA
4
MeL-PPP2CA [nucleoplasm]
(R-HSA-8857791)
p-Y307-PPP2CA [cytosol]
(R-HSA-8857939)
PPP2CA [nucleoplasm]
(R-HSA-165978)
PPP2CA [cytosol]
(R-HSA-165971)
0.593
3
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