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ADRB3 [plasma membrane]
Stable Identifier
R-HSA-390623
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
plasma membrane
Synonyms
Beta-3 adrenoceptor, RecName: Full=Beta-3 adrenergic receptor; AltName: Full=Beta-3 adrenoreceptor; Short=Beta-3 adrenoceptor;
GN Name=ADRB3; Synonyms=ADRB3R, B3AR;
OS Homo sapiens, ADRB3_HUMAN
Locations in the PathwayBrowser
Expand all
Signal Transduction (Homo sapiens)
Signaling by GPCR (Homo sapiens)
GPCR downstream signalling (Homo sapiens)
G alpha (s) signalling events (Homo sapiens)
Liganded Gs-activating GPCR acts as a GEF for Gs (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
Liganded Gs-activating GPCRs bind inactive heterotrimeric Gs (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs:Heterotrimeric G-protein Gs (inactive) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
The Ligand:GPCR:Gs complex dissociates (Homo sapiens)
GPCR:ligand complexes that act on Gs:Heterotrimeric G-protein Gs (active) [plasma membrane] (Homo sapiens)
Ligand:GPCR complexes that activate Gs [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
GPCR ligand binding (Homo sapiens)
Class A/1 (Rhodopsin-like receptors) (Homo sapiens)
Amine ligand-binding receptors (Homo sapiens)
Adrenoceptors (Homo sapiens)
ADRB1 bind ADR,NAd (Homo sapiens)
ADRB1,2,3:β-blockers [plasma membrane] (Homo sapiens)
ADRB1,2,3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
ADRB2 bind ADR,NAd (Homo sapiens)
ADRB1,2,3:β-blockers [plasma membrane] (Homo sapiens)
ADRB1,2,3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
ADRB3 bind ADR,NAd (Homo sapiens)
ADRB1,2,3:β-blockers [plasma membrane] (Homo sapiens)
ADRB1,2,3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
β3-agonists:ADBR3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
β-blockers bind ADRB1,2,3 (Homo sapiens)
ADRB1,2,3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
ADRB1,2,3:β-blockers [plasma membrane] (Homo sapiens)
ADRB1,2,3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
β3-agonists bind ADRB3 (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
β3-agonists:ADBR3 [plasma membrane] (Homo sapiens)
ADRB3 [plasma membrane] (Homo sapiens)
External Reference Information
External Reference
UniProt:P13945 ADRB3
Gene Names
ADRB3, ADRB3R, B3AR
Chain
chain:1-408
Reference Genes
BioGPS Gene:155 ADRB3
COSMIC (genes):ADRB3 ADRB3
CTD Gene:155 ADRB3
dbSNP Gene:155 ADRB3
ENSEMBL:ENSG00000188778 ADRB3
ENSEMBL_homo_sapiens_GENE:ENSG00000188778.6 ADRB3
HGNC:288 ADRB3
KEGG Gene (Homo sapiens):155 ADRB3
Monarch:155 ADRB3
NCBI Gene:155 ADRB3
OMIM:109691 ADRB3
UCSC:P13945 ADRB3
Reference Transcript
RefSeq:NM_000025.2 ADRB3
Other Identifiers
11732428_at
11732429_at
155
17076314
206812_PM_at
206812_at
217303_PM_s_at
217303_s_at
33465_at
4049846
4049847
4049848
4049849
4049850
4049851
4049853
4049854
4049855
8150249
GE79361
GO:0002024
GO:0002025
GO:0003013
GO:0004930
GO:0004935
GO:0004939
GO:0005515
GO:0005886
GO:0005975
GO:0006091
GO:0006112
GO:0007165
GO:0007186
GO:0007187
GO:0007188
GO:0007189
GO:0007190
GO:0009409
GO:0015052
GO:0016020
GO:0023052
GO:0030154
GO:0031649
GO:0031699
GO:0040015
GO:0042755
GO:0042803
GO:0043235
GO:0043410
GO:0050873
GO:0051379
GO:0051380
GO:0060089
GO:0071875
GO:0071880
GO:0120162
HMNXSV003030922
Hs.2549.1.S1_3p_a_at
ILMN_1694007
M29932_s_at
PH_hs_0000338
TC08001140.hg
X70811_at
g4557266_3p_at
g4557266_3p_x_at
Participates
as an input of
ADRB3 bind ADR,NAd (Homo sapiens)
β3-agonists bind ADRB3 (Homo sapiens)
as a component of
β3-agonists:ADBR3 [plasma membrane] (Homo sapiens)
ADRB3:ADR,NAd [plasma membrane] (Homo sapiens)
as a member of
ADRB1,2,3 [plasma membrane] (Homo sapiens)
GPCRs that activate Gs [plasma membrane] (Homo sapiens)
Inferred To
Adrb3 [plasma membrane]
(Mus musculus)
Adrb3 [plasma membrane]
(Rattus norvegicus)
ADRB3 [plasma membrane]
(Bos taurus)
ADRB3 [plasma membrane]
(Canis familiaris)
ADRB3 [plasma membrane]
(Gallus gallus)
ADRB3 [plasma membrane]
(Sus scrofa)
Homologues of ADRB3 [plasma membrane]
(Drosophila melanogaster)
Homologues of ADRB3 [plasma membrane]
(Sus scrofa)
Octbeta1R [plasma membrane]
(Drosophila melanogaster)
Octbeta2R [plasma membrane]
(Drosophila melanogaster)
Octbeta3R [plasma membrane]
(Drosophila melanogaster)
Cross References
RefSeq
NP_000016.1
ZINC - World Drugs
ADRB3_HUMAN
Guide to Pharmacology - Targets
30
OpenTargets
ENSG00000188778
ZINC - FDA approved
ADRB3_HUMAN
ZINC - Substances
ADRB3_HUMAN
ZINC - Biogenic
ADRB3_HUMAN
ZINC target
P13945
PRO
P13945
ZINC - Investigational
ADRB3_HUMAN
ZINC - Metabolites
ADRB3_HUMAN
HPA
ENSG00000188778-ADRB3
GeneCards
P13945
Ensembl
ENSP00000343782
,
ENST00000345060
,
ENSG00000188778
Pharos - Targets
P13945
Orphanet
27551
ZINC - Predictions - Purchasable
ADRB3_HUMAN
HMDB Protein
HMDBP10769
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