20130243 |
Preclinical characterization of the selective JAK1/2 inhibitor INCB018424: therapeutic implications for the treatment of myeloproliferative neoplasms
Li, J,
Quintás-Cardama, A,
Rupar, M,
Manshouri, T,
Kantarjian, H,
Burn, T,
Wen, X,
Lo, Y,
Liu, P,
Verstovsek, S,
Covington, M,
Scherle, PA,
Kelley, J,
Waeltz, P,
Caulder, E,
Shepard, S,
Vaddi, K,
Fridman, JS,
Haley, P,
Li, Y,
Rodgers, JD
|
Blood |
2010 |
23061660 |
Discovery of potent and selective pyrazolopyrimidine janus kinase 2 inhibitors
Chang, C,
Siu, M,
Murray, J,
Sampath, D,
Rawson, T,
Ultsch, M,
Hurley, CA,
Gibbons, P,
Pastor, RM,
Eigenbrot, C,
Zhou, A,
Morris, C,
Barrett, K,
Kenny, JR,
Hanan, EJ,
Flynn, S,
Kulagowski, J,
van Abbema, A,
Blair, WS,
Blaney, J,
Lee, L,
Magnuson, SR,
Lyssikatos, JP
|
J. Med. Chem. |
2012 |
20363976 |
Selective inhibition of JAK1 and JAK2 is efficacious in rodent models of arthritis: preclinical characterization of INCB028050
Favata, MF,
Shi, J,
Yeleswaram, S,
Li, J,
Metcalf, B,
Wen, X,
Scherle, PA,
Thomas, B,
McGee, R,
Collins, R,
Newton, RC,
Burn, TC,
Covington, MB,
Friedman, SM,
Shepard, S,
Haley, PJ,
Vaddi, K,
Hollis, G,
Fridman, JS,
Li, Y,
Rodgers, JD,
Collier, P
|
J. Immunol. |
2010 |