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p-Y342-PTK6 [cytosol]
Stable Identifier
R-HSA-8848007
Type
Protein [EntityWithAccessionedSequence]
Species
Homo sapiens
Compartment
cytosol
Synonyms
p-Y342-BRK
Icon
Locations in the PathwayBrowser
Expand all
Cell Cycle (Homo sapiens)
Cell Cycle, Mitotic (Homo sapiens)
Mitotic G1 phase and G1/S transition (Homo sapiens)
G1 Phase (Homo sapiens)
Cyclin D associated events in G1 (Homo sapiens)
Tyrosine kinases phosphorylate Cip/Kip inhibitors bound to CDK4/6:CCND complexes (Homo sapiens)
(p-Y342-PTK6,p-Y397-LYN,p-Y226,Y393-ABL1,p-Y419-SRC,p-5Y-JAK2) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
G1/S Transition (Homo sapiens)
Cyclin E associated events during G1/S transition (Homo sapiens)
SCF(Skp2)-mediated degradation of p27/p21 (Homo sapiens)
Activated PTK6 binds CDKN1B (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates CDKN1B (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
S Phase (Homo sapiens)
Cyclin A:Cdk2-associated events at S phase entry (Homo sapiens)
SCF(Skp2)-mediated degradation of p27/p21 (Homo sapiens)
Activated PTK6 binds CDKN1B (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates CDKN1B (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
Signal Transduction (Homo sapiens)
Signaling by Non-Receptor Tyrosine Kinases (Homo sapiens)
Signaling by PTK6 (Homo sapiens)
ERBB2 Activates PTK6 Signaling (Homo sapiens)
ERBB2 promotes PTK6 autophosphorylation (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 Activates STAT3 (Homo sapiens)
Activated PTK6 binds STAP2 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates STAP2 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates STAT3 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2:STAT3 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
SOCS3 binds activated PTK6 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:SOCS3 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
STAP2 recruits STAT3 to PTK6 (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2:STAT3 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 Down-Regulation (Homo sapiens)
PTPN1 binds PTK6 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:PTPN1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTPN1 dephosphorylates PTK6 (Homo sapiens)
p-Y342-PTK6:PTPN1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
SRMS phosphorylates PTK6 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 Regulates Cell Cycle (Homo sapiens)
Activated PTK6 binds CDKN1B (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates CDKN1B (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 Regulates Proteins Involved in RNA Processing (Homo sapiens)
PTK6 translocates to the nucleus (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 Regulates RHO GTPases, RAS GTPase and MAP kinases (Homo sapiens)
PTK6 binds ARHGAP35 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:ARHGAP35 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 binds BCAR1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:BCAR1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 binds PXN (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:PXN [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates ARHGAP35 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:ARHGAP35 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates BCAR1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:BCAR1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates PXN (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:PXN [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 Regulates RTKs and Their Effectors AKT1 and DOK1 (Homo sapiens)
PTK6 binds AKT1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:AKT1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 binds ARAP1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:ARAP1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 binds DOK1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:DOK1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates AKT1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:AKT1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y315,Y326-AKT1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates ARAP1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:ARAP1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates CBL (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
PTK6 phosphorylates DOK1 (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
p-Y342-PTK6:DOK1 [cytosol] (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
Signaling by Receptor Tyrosine Kinases (Homo sapiens)
Signaling by ERBB2 (Homo sapiens)
ERBB2 Activates PTK6 Signaling (Homo sapiens)
ERBB2 promotes PTK6 autophosphorylation (Homo sapiens)
p-Y342-PTK6 [cytosol] (Homo sapiens)
External Reference Information
External Reference
UniProt:Q13882 PTK6
Gene Names
PTK6, BRK
Chain
chain:1-451
Reference Genes
BioGPS Gene:5753 PTK6
COSMIC (genes):PTK6 PTK6
CTD Gene:5753 PTK6
dbSNP Gene:5753 PTK6
ENSEMBL:ENSG00000101213 PTK6
HGNC:9617 PTK6
KEGG:hsa:5753 PTK6
Monarch:5753 PTK6
NCBI Gene:5753 PTK6
OMIM:602004 PTK6
UCSC:Q13882 PTK6
Reference Transcript
RefSeq:NM_001256358.1 PTK6
RefSeq:NM_005975.3 PTK6
Other Identifiers
11748835_a_at
11755228_a_at
1208_at
1553114_3p_a_at
1553114_PM_a_at
1553114_a_at
16921268
206482_PM_at
206482_at
33559_at
3913927
3913928
3913929
3913931
3913932
3913933
3913936
3913937
3913938
3913939
3913941
3913942
5753
8067662
A_23_P56978
GE484877
GE80189
GO:0001726
GO:0002376
GO:0003824
GO:0004672
GO:0004713
GO:0004715
GO:0005102
GO:0005515
GO:0005524
GO:0005634
GO:0005654
GO:0005737
GO:0005829
GO:0005886
GO:0006468
GO:0007169
GO:0007260
GO:0010976
GO:0016020
GO:0016477
GO:0016604
GO:0016740
GO:0030154
GO:0038128
GO:0042802
GO:0042995
GO:0043226
GO:0045087
GO:0045740
GO:0045742
GO:0045787
GO:0045926
GO:0046427
GO:0046777
GO:0048870
GO:0060575
GO:0061099
GO:0071300
GO:0098542
GO:0140096
HMNXSV003006584
Hs2.51133.1.S1_3p_x_at
ILMN_1764508
ILMN_2075800
PH_hs_0003525
TC20001033.hg
X78549_at
g5174646_3p_at
Participates
as a component of
p-Y342-PTK6:STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y250-STAP2 [cytosol] (Homo sapiens)
p-Y342-PTK6:SOCS3 [cytosol] (Homo sapiens)
p-Y342-PTK6:PTPN1 [cytosol] (Homo sapiens)
p-Y342-PTK6:CDKN1B:(CDK4:CCND1,(CDK2:CCNE1)) [cytosol] (Homo sapiens)
p-Y342-PTK6:PXN [cytosol] (Homo sapiens)
p-Y342-PTK6:ARHGAP35 [cytosol] (Homo sapiens)
p-Y342-PTK6:BCAR1 [cytosol] (Homo sapiens)
p-Y342-PTK6:AKT1 [cytosol] (Homo sapiens)
p-Y342-PTK6:p-Y315,Y326-AKT1 [cytosol] (Homo sapiens)
p-Y342-PTK6:DOK1 [cytosol] (Homo sapiens)
p-Y342-PTK6:ARAP1 [cytosol] (Homo sapiens)
as an input of
Activated PTK6 binds STAP2 (Homo sapiens)
SOCS3 binds activated PTK6 (Homo sapiens)
SRMS phosphorylates PTK6 (Homo sapiens)
Activated PTK6 binds CDKN1B (Homo sapiens)
PTK6 binds PXN (Homo sapiens)
PTK6 binds ARHGAP35 (Homo sapiens)
PTK6 binds BCAR1 (Homo sapiens)
PTK6 binds AKT1 (Homo sapiens)
PTK6 binds DOK1 (Homo sapiens)
PTK6 binds ARAP1 (Homo sapiens)
PTK6 translocates to the nucleus (Homo sapiens)
PTPN1 binds PTK6 (Homo sapiens)
as an output of
ERBB2 promotes PTK6 autophosphorylation (Homo sapiens)
PTK6 phosphorylates CDKN1B (Homo sapiens)
PTK6 phosphorylates PXN (Homo sapiens)
PTK6 phosphorylates ARHGAP35 (Homo sapiens)
PTK6 phosphorylates BCAR1 (Homo sapiens)
PTK6 phosphorylates ARAP1 (Homo sapiens)
PTK6 phosphorylates DOK1 (Homo sapiens)
as a candidate of
(p-Y342-PTK6,p-Y397-LYN,p-Y226,Y393-ABL1,p-Y419-SRC,p-5Y-JAK2) [cytosol] (Homo sapiens)
Other forms of this molecule
PTK6 [cytosol]
p-Y342-PTK6 [nucleoplasm]
p-Y351-PTK6 [cytosol]
p-Y342,Y447-PTK6 [cytosol]
Inferred To
p-Y342-Ptk6 [cytosol]
(Mus musculus)
Homologues of p-Y342-PTK6 [cytosol]
(Caenorhabditis elegans)
phospho-Ptk6 [cytosol]
(Rattus norvegicus)
phospho-p-Y342-PTK6 [cytosol]
(Bos taurus)
phospho-p-Y342-PTK6 [cytosol]
(Caenorhabditis elegans)
phospho-p-Y342-PTK6 [cytosol]
(Danio rerio)
phospho-p-Y342-PTK6 [cytosol]
(Sus scrofa)
phospho-p-Y342-PTK6 [cytosol]
(Xenopus tropicalis)
Ghost homologue of p-Y342-PTK6 [cytosol]
(Canis familiaris)
Ghost homologue of p-Y342-PTK6 [cytosol]
(Drosophila melanogaster)
Modified Residues
Name
O4'-phospho-L-tyrosine at 342
Coordinate
342
PsiMod Name
O4'-phospho-L-tyrosine [MOD:00048]
PsiMod Definition
A protein modification that effectively converts an L-tyrosine residue to O4'-phospho-L-tyrosine.
Cross References
RefSeq
NP_005966.1
,
NP_001243287.1
ZINC - World Drugs
PTK6_HUMAN
Guide to Pharmacology - Targets
2182
OpenTargets
ENSG00000101213
ENSEMBL
ENSP00000442460
,
ENSP00000217185
,
ENST00000542869
,
ENST00000217185
ZINC - FDA approved
PTK6_HUMAN
ZINC - Substances
PTK6_HUMAN
ZINC - Biogenic
PTK6_HUMAN
ZINC target
Q13882
PRO
Q13882
PDB
1RJA
,
5D7V
,
5DA3
,
6CZ2
,
2KGT
,
5H2U
,
6CZ4
,
6CZ3
ZINC - Investigational
PTK6_HUMAN
HPA
ENSG00000101213-PTK6
Pharos - Targets
Q13882
ZINC - Predictions - Purchasable
PTK6_HUMAN
HMDB Protein
HMDBP01216
Interactors (31)
Accession
#Entities
Entities
Confidence Score
Evidence (IntAct)
UniProt:Q5JST6 EFHC2
0.781
7
UniProt:O00471 EXOC5
2
EXOC5 [cytosol]
(R-HSA-265045)
EXOC5 [cytosol]
(R-HSA-5623383)
0.718
6
UniProt:Q13882 PTK6
5
PTK6 [cytosol]
(R-HSA-8848000)
p-Y342-PTK6 [cytosol]
(R-HSA-8848007)
p-Y342-PTK6 [nucleoplasm]
(R-HSA-8848937)
p-Y351-PTK6 [cytosol]
(R-HSA-8857570)
p-Y342,Y447-PTK6 [cytosol]
(R-HSA-8849103)
0.713
3
UniProt:Q92841 DDX17
2
monoSUMO1-K50-DDX17 [nucleoplasm]
(R-HSA-3900104)
DDX17 [nucleoplasm]
(R-HSA-3900090)
0.666
4
UniProt:Q5VWX1 KHDRBS2
2
KHDRBS2 [nucleoplasm]
(R-HSA-8849028)
p-Y-KHDRBS2 [nucleoplasm]
(R-HSA-8849031)
0.666
4
UniProt:P42858 HTT
1
HTT [nucleoplasm]
(R-HSA-9023590)
0.666
4
UniProt:O14526 FCHO1
1
FCHO1 [cytosol]
(R-HSA-8862257)
0.666
4
UniProt:P23246 SFPQ
3
SFPQ [nucleoplasm]
(R-HSA-3900138)
p-Y-SFPQ [nucleoplasm]
(R-HSA-8849461)
SFPQ [cytosol]
(R-HSA-9635505)
0.632
5
UniProt:P04626 ERBB2
20
ERBB2 G309E [plasma membrane]
(R-HSA-9665342)
ERBB2 G309A [plasma membrane]
(R-HSA-9665349)
ERBB2 S310F [plasma membrane]
(R-HSA-9665350)
ERBB2 S310Y [plasma membrane]
(R-HSA-9665344)
p-6Y-ERBB2 G309A [plasma membrane]
(R-HSA-9665381)
p-6Y-ERBB2 G309E [plasma membrane]
(R-HSA-9665382)
p-6Y-ERBB2 S310F [plasma membrane]
(R-HSA-9665379)
p-6Y-ERBB2 S310Y [plasma membrane]
(R-HSA-9665385)
p-Y-ERBB2 L755P [plasma membrane]
(R-HSA-9654268)
p-Y-ERBB2 I767M [plasma membrane]
(R-HSA-9654303)
p-Y-ERBB2 T798I [plasma membrane]
(R-HSA-9654618)
p-Y-ERBB2 Y772_A775dup [plasma membrane]
(R-HSA-9665652)
p-Y-ERBB2 T862A [plasma membrane]
(R-HSA-9654695)
p-Y-ERBB2 T798M [plasma membrane]
(R-HSA-9654615)
p-Y-ERBB2 H878Y [plasma membrane]
(R-HSA-9654833)
p-Y-ERBB2 V777L [plasma membrane]
(R-HSA-9654401)
p-Y-ERBB2 L755S [plasma membrane]
(R-HSA-9654194)
p-Y-ERBB2 V777E [plasma membrane]
(R-HSA-9654397)
p-Y-ERBB2 V777M [plasma membrane]
(R-HSA-9654398)
p-Y-ERBB2 L755M [plasma membrane]
(R-HSA-9654191)
0.628
4
UniProt:P08238 HSP90AB1
6
HSP90AB1 [lysosomal lumen]
(R-HSA-9622846)
HSP90AB1 [nucleoplasm]
(R-HSA-5082399)
HSP90AB1 [cytosol]
(R-HSA-419617)
HSP90AB1 [secretory granule lumen]
(R-HSA-6801477)
HSP90AB1 [extracellular region]
(R-HSA-6806463)
HSP90AB1 [ficolin-1-rich granule lumen]
(R-HSA-6801491)
0.564
3
UniProt:O00401 WASL
4
p-Y256-WASL [cytosol]
(R-HSA-2197672)
N-WASP [cytosol]
(R-HSA-201873)
WASL [plasma membrane]
(R-HSA-203010)
WASL [endocytic vesicle membrane]
(R-HSA-535012)
0.556
3
UniProt:Q9NQX0 PRDM6
0.556
3
IntAct:EBI-10171584 80125
0.556
3
UniProt:Q08043 ACTN3
1
ACTN3 [cytosol]
(R-HSA-390565)
0.556
3
UniProt:P78337 PITX1
0.556
3
UniProt:Q13239-3 Q132393
0.556
3
UniProt:Q3KP44 ANR55
0.556
3
UniProt:Q13191 CBLB
1
CBLB [cytosol]
(R-HSA-976009)
0.556
3
UniProt:Q9UKT9 IKZF3
0.556
3
UniProt:Q9BYN7 ZN341
0.556
3
UniProt:O14770-4 MEIS2
0.556
3
UniProt:Q5T5P2-6 KIAA1217
0.556
3
UniProt:Q8N9I9 DTX3
0.556
3
UniProt:Q8TDC0 MYOZ3
0.556
3
UniProt:Q04864 REL
2
REL [cytosol]
(R-HSA-1168579)
REL [nucleoplasm]
(R-HSA-1168585)
0.556
3
UniProt:Q13064 MKRN3
0.556
3
UniProt:P17987 TCP1
1
TCP1 [cytosol]
(R-HSA-390448)
0.527
3
UniProt:P50991 CCT4
1
CCT4 [cytosol]
(R-HSA-390458)
0.527
3
UniProt:P50990 CCT8
5
CCT8 [secretory granule lumen]
(R-HSA-6801035)
CCT8 [extracellular region]
(R-HSA-6806238)
CCT8 [azurophil granule lumen]
(R-HSA-6799369)
CCT8 [ficolin-1-rich granule lumen]
(R-HSA-6800894)
CCT8 [cytosol]
(R-HSA-390449)
0.527
3
UniProt:P49368 CCT3
1
CCT3 [cytosol]
(R-HSA-390463)
0.527
3
UniProt:Q16543 CDC37
1
CDC37 [cytosol]
(R-HSA-1221609)
0.499
4
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